Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3',5'-cyclic GMP | - |
Homo sapiens | |
6-mercaptopurine ribonucleotide | - |
Homo sapiens | |
adenosine 3',5'-AMP | - |
Homo sapiens | |
adenylosuccinate | competitive with respect to IMP | Homo sapiens | |
ADP | - |
Homo sapiens | |
AMP | competitive with respect to IMP | Homo sapiens | |
CDP | - |
Homo sapiens | |
CMP | - |
Homo sapiens | |
dAMP | - |
Homo sapiens | |
dCMP | - |
Homo sapiens | |
dGDP | - |
Homo sapiens | |
dGMP | - |
Homo sapiens | |
GDP | competitive with respect to GTP | Homo sapiens | |
GMP | competitive with respect to GTP | Homo sapiens | |
IDP | - |
Homo sapiens | |
succinate | - |
Homo sapiens | |
TDP | - |
Homo sapiens | |
TMP | - |
Homo sapiens | |
UDP | - |
Homo sapiens | |
UMP | - |
Homo sapiens | |
XMP | competitive with respect to IMP | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.031 | - |
GTP | - |
Homo sapiens | |
0.037 | - |
IMP | - |
Homo sapiens | |
0.95 | - |
Asp | - |
Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ba2+ | can replace Mg2+ with lower efficiency | Homo sapiens | |
Ca2+ | can replace Mg2+ with lower efficiency | Homo sapiens | |
Co2+ | can replace Mg2+ with lower efficiency | Homo sapiens | |
Mg2+ | divalent cation required, maximal activity obtained with Mg2+ | Homo sapiens | |
Mn2+ | can replace Mg2+ with lower efficiency | Homo sapiens | |
Ni2+ | can replace Mg2+ with lower efficiency | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
partial | Homo sapiens |
Reaction | Comment | Organism | Reaction ID |
---|---|---|---|
GTP + IMP + L-aspartate = GDP + phosphate + N6-(1,2-dicarboxyethyl)-AMP | sequential rapid equilibrium fully random mechanism | Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
placenta | - |
Homo sapiens | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
0.00641 | - |
- |
Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
GTP + IMP + L-Asp | - |
Homo sapiens | GDP + phosphate + adenylosuccinate | - |
? |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
6.5 | 7.4 | - |
Homo sapiens |