Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 6.2.1.64 extracted from

  • Muraoka, H.; Yoshimura, C.; Kawabata, R.; Tsuji, S.; Hashimoto, A.; Ochiiwa, H.; Nakagawa, F.; Fujioka, Y.; Matsuo, K.; Ohkubo, S.
    Activity of TAS4464, a novel NEDD8 activating enzyme E1 inhibitor, against multiple myeloma via inactivation of nuclear factor ?B pathways (2019), Cancer Sci., 110, 3802-3810 .
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
TAS4464 highly potent inhibitor Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
KMS-11 cell
-
Homo sapiens
-
KMS-12-BM cell
-
Homo sapiens
-
KMS-26 cell
-
Homo sapiens
-
MM1-S cell
-
Homo sapiens
-
multiple myeloma cell
-
Homo sapiens
-

Synonyms

Synonyms Comment Organism
NEDD8 activating enzyme E1
-
Homo sapiens