Crystallization (Comment) | Organism |
---|---|
hanging-drop vapour-diffusion method, CYP-5, X-ray structure solved to a resolution of 1.75 A | Caenorhabditis elegans |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
cyclosporin A | IC50: 50 nM | Caenorhabditis elegans |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
cytoplasm | - |
Caenorhabditis elegans | 5737 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Caenorhabditis elegans | P52014 | the organism expressed 18 cyclophilin isoforms, eight of which are conserved single domain forms, comprising two closely related secreted or type B forms, CYP-5 and CYP-6 | - |
Purification (Comment) | Organism |
---|---|
CYP-5 | Caenorhabditis elegans |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
N-succinyl-Ala-Ala-(trans)-Pro-Phe-4-nitroanilide | - |
Caenorhabditis elegans | N-succinyl-Ala-Ala-(cis)-Pro-Phe-4-nitroanilide | - |
? |
Synonyms | Comment | Organism |
---|---|---|
CYP-5 | - |
Caenorhabditis elegans |
CYP-6 | - |
Caenorhabditis elegans |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00005 | - |
IC50: 50 nM | Caenorhabditis elegans | cyclosporin A |