Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1-[3-(benzhydrylaminocarbonyl)propyl]uracil | 1429fold selectivity over human enzyme | Plasmodium falciparum | |
1-[3-(tritylaminocarbonyl)propyl]uracil | 4545fold selectivity over human enzyme | Plasmodium falciparum |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Plasmodium falciparum | - |
- |
- |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0002 | - |
1-[3-(tritylaminocarbonyl)propyl]uracil | pH 8.0, temperature not specified in the publication | Plasmodium falciparum | |
0.0007 | - |
1-[3-(benzhydrylaminocarbonyl)propyl]uracil | pH 8.0, temperature not specified in the publication | Plasmodium falciparum |