Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 3.5.1.98 extracted from

  • Duong, V.; Bret, C.; Altucci, L.; Mai, A.; Duraffourd, C.; Loubersac, J.; Harmand, P.O.; Bonnet, S.; Valente, S.; Maudelonde, T.; Cavailles, V.; Boulle, N.
    Specific activity of class II histone deacetylases in human breast cancer cells (2008), Mol. Cancer Res., 6, 1908-1919.
    View publication on PubMedView publication on EuropePMC

Cloned(Commentary)

Cloned (Comment) Organism
full-length HDAC1 with COOH-terminal His tag is expressed using baculovirus expression system Homo sapiens
full-length HDAC2 with COOH-terminal His tag is expressed using baculovirus expression system Homo sapiens
full-length HDAC3 with COOH-terminal His tag is expressed using baculovirus expression system Homo sapiens
full-length HDAC4 with COOH-terminal His tag is expressed using baculovirus expression system Homo sapiens
full-length HDAC8 with COOH-terminal His tag is expressed using baculovirus expression system Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
MC1568 specificity for class II HDACs; specificity for class II HDACs; specificity for class II HDACs; specificity for class II HDACs; specificity for class II HDACs Homo sapiens
MC1575 specificity for class II HDACs; specificity for class II HDACs; specificity for class II HDACs; specificity for class II HDACs; specificity for class II HDACs Homo sapiens
suberoylanilide hydroxamic acid SAHA; SAHA; SAHA; SAHA; SAHA Homo sapiens
trichostatin A TSA; TSA; TSA; TSA; TSA Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
cytoplasm depending on phosphorylation status Homo sapiens 5737
-
nucleus depending on phosphorylation status Homo sapiens 5634
-

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Homo sapiens P56524
-
-
Homo sapiens Q13547
-
-
Homo sapiens Q92769
-
-
Homo sapiens Q9BY41
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Homo sapiens

Source Tissue

Source Tissue Comment Organism Textmining
MCF-7 cell
-
Homo sapiens
-

Synonyms

Synonyms Comment Organism
class II histone deacetylase
-
Homo sapiens
HDAC1
-
Homo sapiens
HDAC2
-
Homo sapiens
HDAC3
-
Homo sapiens
HDAC4
-
Homo sapiens
HDAC8
-
Homo sapiens
histone deacetylase
-
Homo sapiens