Cloned (Comment) | Organism |
---|---|
- |
Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(E)-2-((1H-benzo[d]imidazol-2-yl)methylene)-5-propylthiazolidin-4-one | potent small-molecule ADAMTS-5 inhibitor with good permeability | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | Q9UNA0 | - |
- |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00017 | - |
pH 7.5, 37°C | Homo sapiens | (E)-2-((1H-benzo[d]imidazol-2-yl)methylene)-5-propylthiazolidin-4-one | |
0.021 | - |
pH 7.5, 37°C | Homo sapiens | (E)-2-((1H-benzo[d]imidazol-2-yl)methylene)-5-propylthiazolidin-4-one |