Cloned (Comment) | Organism |
---|---|
expressed in Sf9 cells | Mus musculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
QEYKAHHSYKLMS | - |
Mus musculus | |
SC81956 | demonstrates noncompetitive inhibition kinetics | Mus musculus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
aggrecan + H2O | Mus musculus | cleavage at the Glu373-Ala374 site | fragments of aggrecan | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
aggrecan + H2O | cleavage at the Glu373-Ala374 site | Mus musculus | fragments of aggrecan | - |
? | |
K(6-(fluorescein-5-carboxamido)-hexanoic acid)-DVQEFRGVTAVIR-C(QSY9)-KGK + H2O | - |
Mus musculus | C(QSY9) + KGK + K(6-(fluorescein-5-carboxamido)-hexanoic acid)-DVQEFRGVTAVIR | - |
? |
Synonyms | Comment | Organism |
---|---|---|
a disintegrin and metalloproteinase with thrombospondin motifs-4 | - |
Mus musculus |
ADAMTS-4 | - |
Mus musculus |
aggrecanase 1 | - |
Mus musculus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0000228 | - |
SC81956 | at 37°C | Mus musculus | |
0.026 | - |
QEYKAHHSYKLMS | at 37°C | Mus musculus |