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Literature summary for 3.4.24.11 extracted from

  • Malfroy, B.; Schwartz, J.C.
    Properties of enkephalinase from rat kidney: comparison of dipeptidyl-carboxypeptidase and endopeptidase activities (1982), Biochem. Biophys. Res. Commun., 106, 276-285.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
EDTA
-
Mus musculus
EDTA
-
Rattus norvegicus
phosphoramidon
-
Mus musculus
phosphoramidon
-
Rattus norvegicus
thiorphan
-
Mus musculus
thiorphan
-
Rattus norvegicus

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.008
-
Tyr-Gly-Gly-Phe-Met
-
Rattus norvegicus
0.013
-
Tyr-D-Ala-Gly-Phe-Met
-
Rattus norvegicus
0.018
-
Tyr-D-Ala-Gly-Phe-Leu
-
Rattus norvegicus
0.019
-
Tyr-D-Ala-Gly-Phe-Leu
-
Mus musculus
0.061
-
Tyr-D-Ala-Gly-Phe-met-NH2
-
Rattus norvegicus
0.072
-
Tyr-D-Ala-Gly-Phe-met-NH2
-
Mus musculus
0.32
-
Tyr-D-Ala-Gly-Phe-met-NH2
-
Rattus norvegicus
0.35
-
hippuryl-Arg-Arg-Leu-2-naphthylamide
-
Rattus norvegicus
0.38
-
hippuryl-Arg-Arg-Ala-2-naphthylamide
-
Rattus norvegicus

Localization

Localization Comment Organism GeneOntology No. Textmining
membrane bound Rattus norvegicus 16020
-

Metals/Ions

Metals/Ions Comment Organism Structure
additional information metalloproteinase Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
corpus striatum
-
Mus musculus
-
kidney
-
Mus musculus
-
kidney
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
D-Ala2-Leu5-enkephalin + H2O i.e. Tyr-D-Ala-Gly-Phe-Leu Mus musculus Tyr-D-Ala-Gly + Phe-Leu
-
?
D-Ala2-Leu5-enkephalin + H2O i.e. Tyr-D-Ala-Gly-Phe-Leu Rattus norvegicus Tyr-D-Ala-Gly + Phe-Leu
-
?
enkephalin + H2O hydrolysis at Gly3-Phe4 Rattus norvegicus ?
-
?
hippuryl-Arg-Arg-Ala-2-naphthylamide + H2O
-
Rattus norvegicus hippuryl-Arg-Arg + Ala-2-naphthylamide
-
?
hippuryl-Arg-Arg-Leu-2-naphthylamide + H2O
-
Rattus norvegicus hippuryl-Arg-Arg + Leu-2-naphthylamide
-
?
Tyr-D-Ala-Gly-Phe-Met + H2O
-
Rattus norvegicus Tyr-D-Ala-Gly + Phe-Met
-
?
Tyr-D-Ala-Gly-Phe-Met-NH2 + H2O
-
Mus musculus Tyr-D-Ala-Gly + Phe-Met-NH2
-
?
Tyr-D-Ala-Gly-Phe-Met-NH2 + H2O
-
Rattus norvegicus Tyr-D-Ala-Gly + Phe-Met-NH2
-
?
Tyr-Gly-Gly-Phe-Met + H2O i.e. methionine enkephalin Rattus norvegicus Tyr-Gly-Gly + Phe-Met
-
?

Turnover Number [1/s]

Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
6.83
-
hippuryl-Arg-Arg-Ala-2-naphthylamide
-
Rattus norvegicus
17.4
-
Tyr-D-Ala-Gly-Phe-Met
-
Rattus norvegicus
21.1
-
Tyr-Gly-Gly-Phe-Met
-
Rattus norvegicus
42
-
Tyr-D-Ala-Gly-Phe-met-NH2
-
Rattus norvegicus
72
-
hippuryl-Arg-Arg-Leu-2-naphthylamide
-
Rattus norvegicus