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Literature summary for 3.4.24.11 extracted from

  • Morales-Mulia, M.; de Gortari, P.; Amaya, M.I.; Mendez, M.
    Activity and expression of enkephalinase and aminopeptidase N in regions of the mesocorticolimbic system are selectively modified by acute ethanol administration (2012), J. Mol. Neurosci., 46, 58-67.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
thiorphan
-
Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
brain ethanol induces a transitory increase in NEP activities in the frontal cortex and ventral tegmental area, and in the nucleus accumbens Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
N-dansyl-Ala-Gly-D-(4-nitro-Phe)-Gly + H2O
-
Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
enkephalinase
-
Rattus norvegicus
NEP
-
Rattus norvegicus

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.4
-
assay at Rattus norvegicus

Expression

Organism Comment Expression
Rattus norvegicus ethanol induces an increase in NEP mRNA in the frontal cortex up