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Literature summary for 3.4.24.11 extracted from

  • Li, M.; Sun, M.; Liu, Y.; Yu, J.; Yang, H.; Fan, D.; Chui, D.
    Copper downregulates neprilysin activity through modulation of neprilysin degradation (2010), J. Alzheimers Dis., 19, 161-169.
    View publication on PubMed

Cloned(Commentary)

Cloned (Comment) Organism
recombinantly expressed Mus musculus

Inhibitors

Inhibitors Comment Organism Structure
thiorphan
-
Mus musculus

Metals/Ions

Metals/Ions Comment Organism Structure
Cu2+ enzymatic activity is decreased in a dose-and time-dependent manner Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
Neuro-2a cell
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
succinyl-Ala-Ala-Phe-7-amido-4-methylcoumarin + H2O
-
Mus musculus ?
-
?

Synonyms

Synonyms Comment Organism
neprilysin
-
Mus musculus

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Mus musculus

Expression

Organism Comment Expression
Mus musculus decreased expresssion upon treatment with Cu2+ down