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Literature summary for 3.4.23.B8 extracted from

  • Kimura, T.; Nguyen, J.T.; Maegawa, H.; Nishiyama, K.; Arii, Y.; Matsui, Y.; Hayashi, Y.; Kiso, Y.
    Chipping at large, potent human T-cell leukemia virus type 1 protease inhibitors to uncover smaller, equipotent inhibitors (2007), Bioorg. Med. Chem. Lett., 17, 3276-3280.
    View publication on PubMed
Search for more literature for 3.4.23.B8

Inhibitors

Inhibitors Comment Organism Structure
Ac-Ala-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 56% Human T-cell leukemia virus type I
Ac-allophenylnorstatine-Pro-Val-Met-His-OH HTLV-I inhibition below 30% Human T-cell leukemia virus type I
Ac-Gln-(R)-S-methyl-L-cysteine-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 51% Human T-cell leukemia virus type I
Ac-Gln-Ile-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 85% Human T-cell leukemia virus type I
Ac-Gln-Leu-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 54% Human T-cell leukemia virus type I
Ac-Gln-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid- (R)-S-methyl-L-Cys-Met-NH2 HTLV-I inhibition below 30% Human T-cell leukemia virus type I
Ac-Gln-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Ile-Met-NH2 HTLV-I inhibition 74% Human T-cell leukemia virus type I
Ac-Gln-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Leu-Met-NH2 HTLV-I inhibition 30% Human T-cell leukemia virus type I
Ac-Gln-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Thr-Met-NH2 HTLV-I inhibition below 30% Human T-cell leukemia virus type I
Ac-Gln-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 66%; HTLV-I inhibition 99% Human T-cell leukemia virus type I
Ac-Gln-Val-allophenylnorstatine-Pro-Val-Met-His-OH HTLV-I inhibition 49% Human T-cell leukemia virus type I
Ac-Ile-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Ile-Met-NH2 HTLV-I inhibition 94% Human T-cell leukemia virus type I
Ac-Ile-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Gln-NH2 HTLV-I inhibition 86% Human T-cell leukemia virus type I
Ac-Ile-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Ile-NH2 HTLV-I inhibition 78% Human T-cell leukemia virus type I
Ac-Ile-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Leu-NH2 HTLV-I inhibition 54% Human T-cell leukemia virus type I
Ac-Ile-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 87% Human T-cell leukemia virus type I
Ac-Ile-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Phe-NH2 HTLV-I inhibition 84% Human T-cell leukemia virus type I
Ac-Ile-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Val-NH2 HTLV-I inhibition 70% Human T-cell leukemia virus type I
Ac-Leu-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 83% Human T-cell leukemia virus type I
Ac-Phe-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 74% Human T-cell leukemia virus type I
Ac-Val-allophenylnorstatine-Pro-Val-Met-His-OH HTLV-I inhibition below 30% Human T-cell leukemia virus type I
Ac-Val-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-NH2 HTLV-I inhibition 77% Human T-cell leukemia virus type I
H-allophenylnorstatine-Pro-Val-Met-His-OH HTLV-I inhibition below 30% Human T-cell leukemia virus type I
H-Gln-Val-allophenylnorstatine-Pro-Val-Met-His-OH HTLV-I inhibition below 30% Human T-cell leukemia virus type I
H-Pro-Gln-Val-allophenylnorstatine-(R)-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid-Val-Met-His-OH HTLV-I inhibition 99% Human T-cell leukemia virus type I
H-Pro-Gln-Val-allophenylnorstatine-Pro-NH2 HTLV-I inhibition below 30% Human T-cell leukemia virus type I
H-Pro-Gln-Val-allophenylnorstatine-Pro-Val-Met-His-OH HTLV-I inhibition 94% Human T-cell leukemia virus type I
H-Pro-Gln-Val-allophenylnorstatine-Pro-Val-Met-NH2 HTLV-I inhibition 86% Human T-cell leukemia virus type I
H-Pro-Gln-Val-allophenylnorstatine-Pro-Val-NH2 HTLV-I inhibition below 30% Human T-cell leukemia virus type I
H-Val-allophenylnorstatine-Pro-Val-Met-His-OH HTLV-I inhibition below 30% Human T-cell leukemia virus type I

Organism

Organism UniProt Comment Textmining
Human T-cell leukemia virus type I
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-
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Synonyms

Synonyms Comment Organism
HTLV-I protease
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 Human T-cell leukemia virus type I