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Literature summary for 3.4.23.5 extracted from

  • Ollinger, K.
    Inhibition of cathepsin D prevents free-radical-induced apoptosis in rat cardiomyocytes (2000), Arch. Biochem. Biophys., 373, 346-351.
    View publication on PubMed

Application

Application Comment Organism
medicine pretreatment with pepstatin A inhibits apoptosis in cells exposed to naphthazarin (5,8-dihydroxy-1,4-naphthoquinone), naphthazarin releases enzyme from lysosomes to cytosol, later, enzyme reappears in granules of increased size, and activity is restored Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
pepstatin A pretreatment inhibits apoptosis in cells exposed to naphthazarin (5,8-dihydroxy-1,4-naphthoquinone) Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
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-
-

Source Tissue

Source Tissue Comment Organism Textmining
heart cardiomyocyte primary culture Rattus norvegicus
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