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Literature summary for 3.4.23.17 extracted from

  • Azaryan, A.V.; Wong, M.; Friedman, T.C.; Cawley, N.X.; Estivariz, F.E.; Chen, H-C.; Loh, Y.P.
    Purification and characterization of a paired basic residue-specific yeast aspartic protease encoded by the YAP3 gene. Similarity to the mammalian pro-opiomelanocortin-converting enzyme (1993), J. Biol. Chem., 268, 11968-11975.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
DTT 1 mM, stimulates 1.3fold Saccharomyces cerevisiae

Inhibitors

Inhibitors Comment Organism Structure
pepstatin A
-
Saccharomyces cerevisiae

Metals/Ions

Metals/Ions Comment Organism Structure
Ca2+ 5 mM, stimulates Saccharomyces cerevisiae
Ca2+ 1.4fold Saccharomyces cerevisiae

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
68000
-
gel filtration Saccharomyces cerevisiae

Organism

Organism UniProt Comment Textmining
Saccharomyces cerevisiae
-
overexpressing BJ 3501 strain
-
Saccharomyces cerevisiae BJ 3501
-
overexpressing BJ 3501 strain
-

Posttranslational Modification

Posttranslational Modification Comment Organism
glycoprotein
-
Saccharomyces cerevisiae

Purification (Commentary)

Purification (Comment) Organism
overexpressing BJ 3501 strain Saccharomyces cerevisiae

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
Human beta-lipotropin + H2O
-
Saccharomyces cerevisiae More beta-endorphin(1-31) + beta-endorphin(1-29) + beta-endorphin(1-28) + gamma-lipotropin + beta-melanocyte-stimulating hormone ?
Human beta-lipotropin + H2O
-
Saccharomyces cerevisiae BJ 3501 More beta-endorphin(1-31) + beta-endorphin(1-29) + beta-endorphin(1-28) + gamma-lipotropin + beta-melanocyte-stimulating hormone ?
NH2-terminal pro-opiomelanocortin1-77 + H2O
-
Saccharomyces cerevisiae Lys-gamma3-melanotropin + NH2-terminal pro-opiomelanocortin1-49
-
?
NH2-terminal pro-opiomelanocortin1-77 + H2O
-
Saccharomyces cerevisiae BJ 3501 Lys-gamma3-melanotropin + NH2-terminal pro-opiomelanocortin1-49
-
?
Pro-opiomelanocortin + H2O
-
Saccharomyces cerevisiae Adrenocorticotropin + beta-lipotropin
-
?
Pro-opiomelanocortin + H2O
-
Saccharomyces cerevisiae BJ 3501 Adrenocorticotropin + beta-lipotropin
-
?
Small synthetic peptides with paired basic residues + H2O
-
Saccharomyces cerevisiae ?
-
?
Small synthetic peptides with paired basic residues + H2O
-
Saccharomyces cerevisiae BJ 3501 ?
-
?

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
4 4.5
-
Saccharomyces cerevisiae