Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Aaptamine | - |
Staphylococcus aureus | |
berberine chloride | - |
Staphylococcus aureus | |
demethylaaptamine | - |
Staphylococcus aureus | |
demethyloxyaaptamine | - |
Staphylococcus aureus | |
isoaaptamine | the suppression of fibronectin-binding activity by isoaaptamine highlights its potential for the treatment of Staphylococcus aureus infections via inhibition of SrtA activity | Staphylococcus aureus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Staphylococcus aureus | - |
- |
- |
Synonyms | Comment | Organism |
---|---|---|
SrtA | - |
Staphylococcus aureus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
additional information | - |
IC50 for aaptamine is 0.0235 mg/ml, IC50 for isoaaptamine is 0.0037 mg/ml, IC50 for demethylaaptamine is 0.0172 mg/ml, IC50 for demethyloxyaaptamine is 0.0201 mg/ml, IC50 for berberine chloride is 0.0087 mg/ml | Staphylococcus aureus | additional information |