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Literature summary for 3.4.22.63 extracted from

  • Conrad, D.M.; Furlong, S.J.; Doucette, C.D.; West, K.A.; Hoskin, D.W.
    The Ca2+ channel blocker flunarizine induces caspase-10-dependent apoptosis in Jurkat T-leukemia cells (2010), Apoptosis, 15, 597-607.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
benzyloxycarbonyl-AEVD-fluoromethylketone specific caspase-10 inhibitor Homo sapiens
benzyloxycarbonyl-IETD-fluoromethylketone caspase-8/caspase-10 inhibitor Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
JURKAT cell
-
Homo sapiens
-
T-cell leukemia cell
-
Homo sapiens
-

General Information

General Information Comment Organism
physiological function flunarizine triggers apoptosis in Jurkat cells via FADD-independent activation of caspase-10 Homo sapiens