Cloned (Comment) | Organism |
---|---|
- |
Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
acetyl-AEVD-aldehyde | - |
Homo sapiens | |
acetyl-DEVD-aldehyde | - |
Homo sapiens | |
acetyl-IETD-aldehyde | - |
Homo sapiens | |
benzyloxycarbonyl-VAD-fluoromethylketone | t1/2 at 0.001 mM is 98 s | Homo sapiens | |
additional information | KI-values higher than 0.01 mM are determined for acetyl-WEHD-aldehyde and acetyl-YVAD-aldehyde and cowpox serin CrmA | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0000016 | - |
acetyl-DEVD-aldehyde | pH 7.5, 25°C | Homo sapiens | |
0.000425 | - |
acetyl-AEVD-aldehyde | pH 7.5, 25°C | Homo sapiens | |
0.00328 | - |
acetyl-IETD-aldehyde | pH 7.5, 25°C | Homo sapiens |