Inhibitors | Comment | Organism | Structure |
---|---|---|---|
CA-030 | and derivatives | Homo sapiens | |
CA-074 | and derivatives | Homo sapiens | |
E-64 | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P07858 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Abz-Ala-Phe-Arg-Ser-Ala-X-Gln-EDDnp + H2O | kcat/Km for Abz-Ala-Phe-Arg-Ser-Ala-X-Gln-EDDnp, with X is Asn > Tyr, His, Leu, Trp > Ser, Phe, Pro Lys > Asp, Ala | Homo sapiens | Abz-Ala-Phe-Arg + Ser-Ala-X-Gln-EDDnp | - |
? | |
Abz-Ala-Phe-Arg-Ser-X-Arg-Ser-Ala-Gln-EDDnp + H2O | kcat/Km for Abz-Ala-Phe-Arg-Ser-X-Arg-Ser-Ala-Gln-EDDnp, with X is Asn > Trp, Tyr, Ala > Ser, Phe > His, Lys > Asp, Leu, Pro | Homo sapiens | Abz-Ala-Phe-Arg + Ser-X-Arg-Ser-Ala-Gln-EDDnp | - |
? | |
Abz-Ala-X-Ala-Phe-Arg-Ser-Ala-Gln-EDDnp + H2O | kcat/Km for Abz-Ala-X-Ala-Phe-Arg-Ser-Ala-Gln-EDDnp, with X is Leu, Tyr > Phe, Ala, Ser, Pro > His, Lys > Asn, Asp | Homo sapiens | Abz-Ala-X-Ala-Phe-Arg + Ser-Ala-Gln-EDDnp | - |
? | |
Abz-Ala-X-Arg-Ser-Ala-Ala-Gln-EDDnp + H2O | kcat/Km for Abz-Ala-X-Arg-Ser-Ala-Ala-Gln-EDDnp, with X is Phe, Leu > Arg > Ala > Pro | Homo sapiens | Abz-Ala-X-Arg + Ser-Ala-Ala-Gln-EDDnp | - |
? | |
Abz-X-Ala-Phe-Arg-Ser-Ala-Gln-EDDnp + H2O | kcat/Km for Abz-X-Ala-Phe-Arg-Ser-Ala-Gln-EDDnp, with X is Leu, Phe, Trp > Ser, Asn, Asp, Ala > Tyr, His, Lys | Homo sapiens | Abz-X-Ala-Phe-Arg + Ser-Ala-Gln-EDDnp | - |
? | |
benzyloxycarbonyl-Phe-Arg-AMC + H2O | - |
Homo sapiens | ? | - |
? | |
Dnp-Gly-Phe-Arg-Trp-X-OH + H2O | kcat/Km for Dnp-Gly-Phe-Arg-Trp-X-OH, with X is Phe > Tyr, Ile > Leu > Cval > Arg > Lys, Pro > Gln, Ser > Asp, Glu, Ala | Homo sapiens | Dnp-Gly-Phe + Arg-Trp-X-OH | - |
? | |
Dnp-Gly-Phe-Arg-X-Trp-OH + H2O | kcat/Km for Dnp-Gly-Phe-Arg-X-Trp-OH, with X is Phe > Ser > Leu > Ala > Ile > Tyr, Val > Gln > Lys > Gly > His, Asp > Arg > Glu | Homo sapiens | Dnp-Gly-Phe + Arg-X-Trp-OH | - |
? | |
Dnp-Gly-Phe-X-Phe-Trp-OH + H2O | kcat/Km for Dnp-Gly-Phe-X-Phe-Trp-OH, with X is Arg > Lys > Phe > Leu > Val > His, Gln > Ser > Gly Ala > Glu > Tyr > Ile, Asp | Homo sapiens | Dnp-Gly-Phe-X + Phe-Trp-OH | - |
? | |
Dnp-Gly-X-Arg-Phe-Trp-OH + H2O | kcat/Km for Dnp-Gly-X-Arg-Phe-Trp-OH, with X is Phe > Tyr > Lys > Val > Ala > Ile > Ser, Pro > His > Leu > Arg > Asp, Glu | Homo sapiens | Dnp-Gly-X-Arg + Phe-Trp-OH | - |
? | |
additional information | active site mapping with peptidic substrates and inhibitors | Homo sapiens | ? | - |
? |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00000224 | - |
pH and temperature not specified in the publication | Homo sapiens | CA-074 | |
0.00000228 | - |
pH and temperature not specified in the publication | Homo sapiens | CA-030 |
kcat/KM Value [1/mMs-1] | kcat/KM Value Maximum [1/mMs-1] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
Abz-Ala-Phe-Arg-Ser-Ala-X-Gln-EDDnp | kcat/Km for Abz-Ala-Phe-Arg-Ser-Ala-X-Gln-EDDnp: Asn > Tyr, His, Leu, Trp > Ser, Phe, Pro Lys > Asp, Ala | Homo sapiens | |
additional information | - |
Abz-Ala-Phe-Arg-Ser-X-Arg-Ser-Ala-Gln-EDDnp | kcat/Km for Abz-Ala-Phe-Arg-Ser-X-Arg-Ser-Ala-Gln-EDDnp: Asn > Trp, Tyr, Ala > Ser, Phe > His, Lys > Asp, Leu, Pro | Homo sapiens | |
additional information | - |
Abz-Ala-X-Arg-Ser-Ala-Ala-Gln-EDDnp | kcat/Km for Abz-Ala-X-Arg-Ser-Ala-Ala-Gln-EDDnp: Phe, Leu > Arg > Ala > Pro | Homo sapiens | |
additional information | - |
Abz-Ala-X-Ala-Phe-Arg-Ser-Ala-Gln-EDDnp | kcat/Km for Abz-Ala_X-Ala-Phe-Arg-Ser-Ala-Gln-EDDnp: Leu, Tyr > Phe, Ala, Ser, Pro > His, Lys > Asn, Asp | Homo sapiens | |
additional information | - |
Abz-X-Ala-Phe-Arg-Ser-Ala-Gln-EDDnp | kcat/Km for Abz-X-Ala-Phe-Arg-Ser-Ala-Gln-EDDnp: Leu, Phe, Trp > Ser, Asn, Asp, Ala > Tyr, His, Lys | Homo sapiens | |
additional information | - |
Dnp-Gly-Phe-Arg-Trp-X-OH | kcat/Km for Dnp-Gly-Phe-Arg-Trp-X-OH: Phe > Tyr, Ile > Leu > Cval > Arg > Lys, Pro > Gln, Ser > Asp, Glu, Ala | Homo sapiens | |
additional information | - |
Dnp-Gly-Phe-Arg-X-Trp-OH | kcat/Km for Dnp-Gly-Phe-Arg-X-Trp-OH: Phe > Ser > Leu > Ala > Ile > Tyr, Val > Gln > Lys > Gly > His, Asp > Arg > Glu | Homo sapiens | |
additional information | - |
Dnp-Gly-Phe-X-Phe-Trp-OH | kcat/Km for Dnp-Gly-Phe-X-Phe-Trp-OH: Arg > Lys > Phe > Leu > Val > His, Gln > Ser > Gly Ala > Glu > Tyr > Ile, Asp | Homo sapiens | |
additional information | - |
Dnp-Gly-X-Arg-Phe-Trp-OH | kcat/Km for Dnp-Gly-X-Arg-Phe-Trp-OH: Phe > Tyr > Lys > Val > Ala > Ile > Ser, Pro > His > Leu > Arg > Asp, Glu | Homo sapiens |