Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Abz-Phe-Arg-Lys-Gln-EDDnp | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00036 | - |
Abz-Leu-Leu-Ala-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Lys-Lys-Met-Asp-Glu-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.0012 | - |
Abz-Lys-Leu-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.0017 | - |
Abz-Arg-Thr-Ser-Arg-Arg-Lys-Arg-Tyr-Ala-Glu-His-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.0018 | - |
Abz-Asp-Met-Ser-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Arg-Ser-Leu-Lys-Arg-Ser-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.0026 | - |
Abz-Lys-Leu-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.004 | - |
benzoyl-Ala-Arg-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
0.0046 | - |
Abz-Glu-Glu-Val-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Arg-Gly-Leu-Lys-Arg-Ser-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.0074 | - |
Abz-Thr-His-Arg-Ser-Lys-Arg-Ser-Ser-Ser-His-Pro-Ile-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.014 | - |
Abz-Ser-Met-Arg-Val-Arg-Arg-His-Ser-Asp-Pro-Ala-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.017 | - |
Abz-Lys-Leu-Arg-Arg-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.021 | - |
Abz-Asp-Tyr-Gln-Lys-Arg-Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Phe-Ala-Glu-Ala-Leu-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.023 | - |
Abz-Phe-Arg-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.023 | - |
benzoyl-Ala-Lys-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
0.025 | - |
Abz-Lys-Lys-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.026 | - |
benzyloxycarbonyl-Arg-Arg-7-amido-4-methylcoumarin | pH 7.5, 37°C | Homo sapiens | |
0.027 | - |
Abz-Lys-Arg-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.043 | - |
Abz-Phe-Arg-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.047 | - |
benzoyl-Ala-Phe-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
0.053 | - |
Abz-Ala-Arg-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.055 | - |
Lys-Ala-Arg-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
0.073 | - |
Abz-Ala-Arg-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.076 | - |
Abz-Ala-Lys-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | Q92876 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
central nervous system | highly expressed in the central nervous system and with elevated level in demyelinating disease | Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Abz-Ala-Arg-Arg-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Ala-Arg + Args-Gln-EDDnp | - |
? | |
Abz-Ala-Arg-Lys-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Ala-Arg + Lys-Gln-EDDnp | - |
? | |
Abz-Ala-Lys-Arg-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Ala-Lys-Arg + Gln-EDDnp | - |
? | |
Abz-Ala-Pro-Ala-Asn-Arg-Ser-Arg-Arg-Gly-Val-Ser-Glu-Thr-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Ala-Pro-Ala-Asn-Arg-Ser-Arg + Arg-Gly-Val-Ser-Glu-Thr-Gln-EDDnp | - |
? | |
Abz-Arg-Thr-Ser-Arg-Arg-Lys-Arg-Tyr-Ala-Glu-His-Lys-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Arg-Thr-Ser-Arg-Arg-Lys-Arg + Tyr-Ala-Glu-His-Lys-Gln-EDDnp | - |
? | |
Abz-Asp-Met-Ser-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Arg-Ser-Leu-Lys-Arg-Ser-Gln-EDDnp + H2O | cleavage sites: Abz-Asp-Met-Ser-Lys-Arg-/-Tyr-Gly-Gly-Phe-Met-Arg-/-Ser-Leu-Lys-Arg-Ser-Gln-EDDnp | Homo sapiens | ? | - |
? | |
Abz-Asp-Tyr-Gln-Lys-Arg-Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Phe-Ala-Glu-Ala-Leu-Gln-EDDnp + H2O | cleavage sites: Abz-Asp-Tyr-Gln-Lys-Arg-/-Tyr-Gly-Gly-Phe-Leu-Lys-Arg-/-Phe-Ala-Glu-Ala-Leu-Gln-EDDnp | Homo sapiens | ? | - |
? | |
Abz-Glu-Glu-Val-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Arg-Gly-Leu-Lys-Arg-Ser-Gln-EDDnp + H2O | cleavage sites: Abz-Glu-Glu-Val-Lys-Arg-/-Tyr-Gly-Gly-Phe-Met-Arg-/-Gly-Leu-Lys-Arg-Ser-Gln-EDDnp | Homo sapiens | ? | - |
? | |
Abz-Leu-Leu-Ala-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Lys-Lys-Met-Asp-Glu-Gln-EDDnp + H2O | cleavage sites: Abz-Leu-Leu-Ala-Lys-Arg-/-Tyr-Gly-Gly-Phe-Met-Lys-Arg-/-Tyr-Gly-Gly-Phe-Met-Lys-/-Lys-Met-Asp-Glu-Gln-EDDnp | Homo sapiens | ? | - |
? | |
Abz-Lys-Arg-Arg-Ser-Ser-Lys-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Lys-Arg-Arg + Ser-Ser-Lys-Gln-EDDnp | - |
? | |
Abz-Lys-Leu-Arg-Arg-Ser-Lys-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Lys-Leu-Arg + Arg-Ser-Lys-Gln-EDDnp + Abz-Lys-Leu-Arg-Arg + Ser-Lys-Gln-EDDnp | - |
? | |
Abz-Lys-Leu-Arg-Ser-Ser-Lys-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Lys-Leu-Arg + Ser-Ser-Lys-Gln-EDDnp | - |
? | |
Abz-Lys-Lys-Arg-Ser-Ser-Lys-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Lys-Lys-Arg + Ser-Ser-Lys-Gln-EDDnp | - |
? | |
Abz-Phe-Arg-Arg-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Phe-Arg + Arg-Gln-EDDnp | - |
? | |
Abz-Phe-Arg-Lys-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Phe-Arg + Lys-Gln-EDDnp | - |
? | |
Abz-Ser-Met-Arg-Val-Arg-Arg-His-Ser-Asp-Pro-Ala-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Ser-Met-Arg-Val-Arg + Arg-His-Ser-Asp-Pro-Ala-Gln-EDDnp | - |
? | |
Abz-Thr-His-Arg-Ser-Lys-Arg-Ser-Ser-Ser-His-Pro-Ile-Gln-EDDnp + H2O | - |
Homo sapiens | Abz-Thr-His-Arg-Ser-Lys-Arg + Ser-Ser-Ser-His-Pro-Ile-Gln-EDDnp | - |
? | |
benzoyl-Ala-Arg-Arg-7-amido-4-carbamoylmethylcoumarin + H2O | - |
Homo sapiens | benzoyl-Ala-Arg + Arg-7-amido-4-carbamoylmethylcoumarin | - |
? | |
benzoyl-Ala-Lys-Arg-7-amido-4-carbamoylmethylcoumarin + H2O | - |
Homo sapiens | benzoyl-Ala-Lys + Arg-7-amido-4-carbamoylmethylcoumarin | - |
? | |
benzoyl-Ala-Phe-Arg-7-amido-4-carbamoylmethylcoumarin + H2O | - |
Homo sapiens | benzoyl-Ala-Phe + Arg-7-amido-4-carbamoylmethylcoumarin | - |
? | |
benzyloxycarbonyl-Arg-Arg-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | benzoyl-Arg + Arg-7-amido-4-methylcoumarin | - |
? | |
human ionotropic glutamate receptor subunit + H2O | - |
Homo sapiens | ? | - |
? | |
human MMP-14 + H2O | - |
Homo sapiens | ? | - |
? | |
Lys-Ala-Arg-Arg-7-amido-4-carbamoylmethylcoumarin + H2O | - |
Homo sapiens | Lys-Ala-Arg + Arg-7-amido-4-carbamoylmethylcoumarin | - |
? | |
myelin basic protein + H2O | - |
Homo sapiens | ? | - |
? | |
nerve growth factor + H2O | - |
Homo sapiens | ? | - |
? | |
neurotrophin-3 + H2O | - |
Homo sapiens | ? | - |
? | |
neurotrophin-4 + H2O | - |
Homo sapiens | ? | - |
? | |
Proenkephalin + H2O | - |
Homo sapiens | Enkephalin + ? | - |
? | |
protein activator receptor + H2O | - |
Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
kallikrein-related peptidase 6 | - |
Homo sapiens |
KLK6 | - |
Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.04 | - |
Abz-Ala-Arg-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.06 | - |
Abz-Asp-Met-Ser-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Arg-Ser-Leu-Lys-Arg-Ser-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.07 | - |
Abz-Arg-Thr-Ser-Arg-Arg-Lys-Arg-Tyr-Ala-Glu-His-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.08 | - |
Abz-Leu-Leu-Ala-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Lys-Lys-Met-Asp-Glu-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.08 | - |
Abz-Glu-Glu-Val-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Arg-Gly-Leu-Lys-Arg-Ser-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.09 | - |
Abz-Phe-Arg-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.1 | - |
Abz-Ser-Met-Arg-Val-Arg-Arg-His-Ser-Asp-Pro-Ala-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.18 | - |
Abz-Asp-Tyr-Gln-Lys-Arg-Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Phe-Ala-Glu-Ala-Leu-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
0.2 | - |
Abz-Thr-His-Arg-Ser-Lys-Arg-Ser-Ser-Ser-His-Pro-Ile-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
1.5 | - |
Abz-Lys-Leu-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
1.95 | - |
Abz-Ala-Lys-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
2 | - |
Abz-Ala-Arg-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
2.4 | - |
Abz-Lys-Leu-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
2.5 | - |
benzoyl-Ala-Lys-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
3 | - |
Abz-Phe-Arg-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
4.6 | - |
Abz-Lys-Arg-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
6.5 | - |
benzyloxycarbonyl-Arg-Arg-7-amido-4-methylcoumarin | pH 7.5, 37°C | Homo sapiens | |
8 | - |
benzoyl-Ala-Arg-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
9 | - |
Abz-Lys-Leu-Arg-Arg-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
9.7 | - |
Lys-Ala-Arg-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
10 | - |
benzoyl-Ala-Phe-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
18 | - |
Abz-Lys-Lys-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.031 | - |
Abz-Phe-Arg-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens |
kcat/KM Value [1/mMs-1] | kcat/KM Value Maximum [1/mMs-1] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.72 | - |
Abz-Ala-Arg-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
3.8 | - |
Abz-Phe-Arg-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
7 | - |
Abz-Ser-Met-Arg-Val-Arg-Arg-His-Ser-Asp-Pro-Ala-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
8.6 | - |
Abz-Asp-Tyr-Gln-Lys-Arg-Tyr-Gly-Gly-Phe-Leu-Lys-Arg-Phe-Ala-Glu-Ala-Leu-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
16 | - |
Abz-Glu-Glu-Val-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Arg-Gly-Leu-Lys-Arg-Ser-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
26 | - |
Abz-Ala-Lys-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
27 | - |
Abz-Ala-Arg-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
27 | - |
Abz-Thr-His-Arg-Ser-Lys-Arg-Ser-Ser-Ser-His-Pro-Ile-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
33 | - |
Abz-Asp-Met-Ser-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Arg-Ser-Leu-Lys-Arg-Ser-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
41 | - |
Abz-Arg-Thr-Ser-Arg-Arg-Lys-Arg-Tyr-Ala-Glu-His-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
70 | - |
Abz-Phe-Arg-Arg-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
107 | - |
benzoyl-Ala-Lys-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
170 | - |
Abz-Lys-Arg-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
190 | - |
Lys-Ala-Arg-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
210 | - |
benzoyl-Ala-Phe-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens | |
228 | - |
Abz-Leu-Leu-Ala-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Lys-Arg-Tyr-Gly-Gly-Phe-Met-Lys-Lys-Met-Asp-Glu-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
250 | - |
benzyloxycarbonyl-Arg-Arg-7-amido-4-methylcoumarin | pH 7.5, 37°C | Homo sapiens | |
529 | - |
Abz-Lys-Leu-Arg-Arg-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
570 | - |
Abz-Lys-Leu-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
720 | - |
Abz-Lys-Lys-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
1983 | - |
Abz-Lys-Leu-Arg-Ser-Ser-Lys-Gln-EDDnp | pH 7.5, 37°C | Homo sapiens | |
2000 | - |
benzoyl-Ala-Arg-Arg-7-amido-4-carbamoylmethylcoumarin | pH 7.5, 37°C | Homo sapiens |