Protein Variants | Comment | Organism |
---|---|---|
H51A | less than 1% of wild-type activity, no autolytic conversion into mature enzyme | West Nile virus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
alpha1-anitrypsin | - |
West Nile virus | |
Aprotinin | - |
West Nile virus | |
deca-D-Arg-NH2 | - |
West Nile virus | |
dodeca-D-Arg-NH2 | - |
West Nile virus | |
dodeka-D-Arg-NH2 | - |
West Nile virus | |
hepta-D-Arg-NH2 | - |
West Nile virus | |
hexa-D-Arg-NH2 | - |
West Nile virus | |
nona-D-Arg-NH2 | reduces infection in primary neurons | West Nile virus | |
octa-D-Arg-NH2 | - |
West Nile virus | |
undeca-D-Arg-NH2 | - |
West Nile virus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.041 | - |
Boc-RVRR-7-amido-4-methylcoumarin | pH 8.0, 18°C | West Nile virus | |
0.043 | - |
Pyr-RTKR-7-amido-4-methylcoumarin | pH 8.0, 18°C | West Nile virus | |
0.146 | - |
Z-RR-7-amido-4-methylcoumarin | pH 8.0, 18°C | West Nile virus |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
30000 | - |
x * 30000, mature protein, SDS-PAGE | West Nile virus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
West Nile virus | - |
recombinantenzyme | - |
Posttranslational Modification | Comment | Organism |
---|---|---|
proteolytic modification | autolytic conversion of 36 kDa NS2B-NS3 construct into the 30 kDa NS3 enzyme | West Nile virus |
Purification (Comment) | Organism |
---|---|
recombinant protein, autolytic conversion of 36 kDa NS2B-NS3 construct into the 30 kDa NS3 enzyme | West Nile virus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Boc-RVRR-7-amido-4-methylcoumarin + H2O | - |
West Nile virus | ? | - |
? | |
additional information | no substrate: Boc-AGPR-AMC, Boc-QAR-AMC, Boc-O-benzyl-EGR-pNA | West Nile virus | ? | - |
? | |
myelin basic protein + H2O | - |
West Nile virus | ? | - |
? | |
Pyr-RTKR-7-amido-4-methylcoumarin + H2O | - |
West Nile virus | ? | - |
? | |
Z-RR-7-amido-4-methylcoumarin + H2O | - |
West Nile virus | ? | - |
? |
Subunits | Comment | Organism |
---|---|---|
? | x * 30000, mature protein, SDS-PAGE | West Nile virus |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.062 | - |
Z-RR-7-amido-4-methylcoumarin | pH 8.0, 18°C | West Nile virus | |
0.073 | - |
Boc-RVRR-7-amido-4-methylcoumarin | pH 8.0, 18°C | West Nile virus | |
43 | - |
Pyr-RTKR-7-amido-4-methylcoumarin | pH 8.0, 18°C | West Nile virus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000001 | - |
undeca-D-Arg-NH2 | pH 8.0, 18°C | West Nile virus | |
0.000001 | - |
dodeka-D-Arg-NH2 | pH 8.0, 18°C | West Nile virus | |
0.000002 | - |
deca-D-Arg-NH2 | pH 8.0, 18°C | West Nile virus | |
0.000006 | - |
nona-D-Arg-NH2 | pH 8.0, 18°C | West Nile virus | |
0.000017 | - |
octa-D-Arg-NH2 | pH 8.0, 18°C | West Nile virus | |
0.000026 | - |
Aprotinin | pH 8.0, 18°C | West Nile virus | |
0.000041 | - |
hepta-D-Arg-NH2 | pH 8.0, 18°C | West Nile virus | |
0.000478 | - |
hexa-D-Arg-NH2 | pH 8.0, 18°C | West Nile virus | |
0.00059 | - |
alpha1-antitrypsin | pH 8.0, 18°C | West Nile virus |