Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Ca2+ | slight inhibition of substrates with one or two Asp/Glu residues at P2-P3 positions | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.16 | - |
GD4KF(NO2)G | 50 mM Ca2+, pH 8.0, 37°C | Homo sapiens | |
0.2 | - |
glycyl-tetra-L-aspartyl-L-lysine beta-naphthylamide | 50 mM Ca2+, pH 8.0, 37°C | Homo sapiens | |
0.525 | - |
glycyl-tetra-L-aspartyl-L-lysine beta-naphthylamide | pH 8.0, 37°C | Homo sapiens | |
596 | - |
N-alpha-benzyloxycarbonyl-L-lysine thiobenzyl ester + | 37°C, pH 8.0 | Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ca2+ | 50 mM, 3fold activation of hydrolysis of substrates of the general type GD4KX | Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
Trypsinogen + H2O | Homo sapiens | - |
? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
G5DKF(NO2)G + H2O | - |
Homo sapiens | ? | - |
? | |
GD4KF(NO2)G + H2O | - |
Homo sapiens | ? | - |
? | |
glycyl-tetra-L-aspartyl-L-lysine beta-naphthylamide + H2O | - |
Homo sapiens | glycyl-tetra-L-aspartyl-L-lysine + beta-naphthylamine | - |
? | |
LTAEEKA + H2O | - |
Homo sapiens | ? | - |
? | |
LTAEEKAAV + H2O | - |
Homo sapiens | ? | - |
? | |
N-alpha-benzyloxycarbonyl-L-lysine thiobenzyl ester + H2O | - |
Homo sapiens | N-alpha-benzyloxycarbonyl-L-lysine + benzylmercaptane | - |
? | |
N-alpha-benzyloxycarbonyl-L-lysine thiobenzyl ester + H2O | - |
Homo sapiens | N-alpha-benzyloxycarbonyl-L-lysine + phenylmethanethiol | - |
? | |
Trypsinogen + H2O | - |
Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
EP 118-1035 | - |
Homo sapiens |
natural enteropeptidase | - |
Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.07 | - |
LTAEEKA | pH 8.0, 37°C | Homo sapiens | |
0.97 | - |
G5DKF(NO2)G | 50 mM Ca2+, pH 8.0, 37°C | Homo sapiens | |
0.97 | - |
glycyl-tetra-L-aspartyl-L-lysine beta-naphthylamide | 50 mM Ca2+, pH 8.0, 37°C | Homo sapiens | |
0.99 | - |
GD4KF(NO2)G | 50 mM Ca2+, pH 8.0, 37°C | Homo sapiens | |
16.67 | - |
glycyl-tetra-L-aspartyl-L-lysine beta-naphthylamide | 50 mM Ca2+, pH 8.0, 37°C | Homo sapiens | |
17.33 | - |
G5DKF(NO2)G | 50 mM Ca2+, pH 8.0, 37°C | Homo sapiens | |
17.83 | - |
GD4KF(NO2)G | 50 mM Ca2+, pH 8.0, 37°C | Homo sapiens | |
21.5 | - |
glycyl-tetra-L-aspartyl-L-lysine beta-naphthylamide | pH 8.0, 37°C | Homo sapiens | |
111 | - |
N-alpha-benzyloxycarbonyl-L-lysine thiobenzyl ester | 37°C, pH 8.0 | Homo sapiens |