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Literature summary for 3.4.21.78 extracted from

  • Bell, J.K.; Goetz, D.H.; Mahrus, S.; Harris, J.L.; Fletterick, R.J.; Craik, C.S.
    The oligomeric structure of human granzyme A is a determinant of its extended substrate specificity (2003), Nat. Struct. Biol., 10, 527-534.
    View publication on PubMed

Cloned(Commentary)

Cloned (Comment) Organism
cDNA subcloned into the yeast vector pPICzalphaA and heterologously expressed in Pichia pastoris Homo sapiens

Crystallization (Commentary)

Crystallization (Comment) Organism
-
Homo sapiens

Protein Variants

Protein Variants Comment Organism
N153Q molecular replacement Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
additional information ecotin has no effect Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Homo sapiens cell death-inducing serine protease ?
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
human
-

Purification (Commentary)

Purification (Comment) Organism
recombinant enzyme Homo sapiens

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information cell death-inducing serine protease Homo sapiens ?
-
?
PSSCL + H2O
-
Homo sapiens Pro-Ser + Ser-Lys-Lys
-
?

Subunits

Subunits Comment Organism
dimer only granzyme that forms a disulfide-linked homodimer Homo sapiens
oligomer
-
Homo sapiens

Synonyms

Synonyms Comment Organism
Gzma
-
Homo sapiens