Inhibitors | Comment | Organism | Structure |
---|---|---|---|
antithrombin | - |
Bos taurus | |
glycosaminoglycan AD17 | - |
Bos taurus | |
glycosaminoglycan AD4 | shows only small inhibitory activity toward thrombin and the inhibition does not proceed beyond 40% inhibition | Bos taurus | |
glycosaminoglycan AD9 | shows only small inhibitory activity toward thrombin and the inhibition does not proceed beyond 40% inhibition | Bos taurus | |
glycosaminoglycan AE11 | modest inhibitory effect on thrombin activity | Bos taurus | |
glycosaminoglycan AE15 | - |
Bos taurus | |
glycosaminoglycan AE29 | - |
Bos taurus | |
glycosaminoglycan AE6 | modest inhibitory effect on thrombin activity | Bos taurus | |
glycosaminoglycan CS-D | - |
Bos taurus | |
glycosaminoglycan CS-E | - |
Bos taurus | |
glycosaminoglycan DE17 | - |
Bos taurus | |
glycosaminoglycan DE2 | - |
Bos taurus | |
glycosaminoglycan DE9 | - |
Bos taurus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
fibrinogen + H2O | Bos taurus | - |
fibrin + fibrinopeptide A + fibrinopeptide B | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
fibrinogen + H2O | - |
Bos taurus | fibrin + fibrinopeptide A + fibrinopeptide B | - |
? |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0001 | - |
- |
Bos taurus | glycosaminoglycan CS-E | |
0.00015 | - |
- |
Bos taurus | glycosaminoglycan DE17 | |
0.00025 | - |
- |
Bos taurus | glycosaminoglycan DE9 | |
0.00055 | - |
- |
Bos taurus | glycosaminoglycan DE2 | |
0.0007 | - |
- |
Bos taurus | glycosaminoglycan AD17 | |
0.00092 | - |
- |
Bos taurus | glycosaminoglycan AE29 | |
0.00095 | - |
- |
Bos taurus | glycosaminoglycan CS-D | |
0.0025 | - |
- |
Bos taurus | glycosaminoglycan AE15 | |
0.00429 | - |
IC50 above 0.00429 mM | Bos taurus | glycosaminoglycan AE6 | |
0.00429 | - |
IC50 above 0.00429 mM | Bos taurus | glycosaminoglycan AE11 | |
0.00429 | - |
IC50 above 0.00429 mM | Bos taurus | glycosaminoglycan AD4 | |
0.00429 | - |
IC50 above 0.00429 mM | Bos taurus | glycosaminoglycan AD9 |