KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
2-[5-Amino-2-(4-fluoro-phenyl)-6-oxo-6H-pyrimidin-1-yl]-N-(1-benzyl-2-oxo-2-thiazol-2-yl-ethyl)-acetamide | K0.5-values | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
2-aminobenzoyl-Gly-Leu-Gln-Arg-Ala-Leu-Glu-Ile-Lys(dinitrophenyl)-NH2 + H2O | - |
Homo sapiens | 2-aminobenzoyl-Gly-Leu-Gln-Arg + Ala-Leu-Glu-Ile-Lys(dinitrophenyl)-NH2 | - |
? | |
2-aminobenzoyl-Ser-Leu-Gly-Arg-Lys-Ile-Gln-Ile-Lys(dinitrophenyl)-NH2 + H2O | - |
Homo sapiens | 2-aminobenzoyl-Ser-Leu-Gly-Arg + Lys-Ile-Gln-Ile-Lys(dinitrophenyl)-NH2 | - |
? | |
benzyloxycarbonyl-Gly-Leu-Gln-Arg-4-methylcoumaryl-7-amide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Gly-Leu-Gln-Arg + 7-amino-4-methylcoumarin | - |
? | |
benzyloxycarbonyl-Ser-Leu-Gly-Arg-4-methylcoumaryl-7-amide + H2O | - |
Homo sapiens | benzyloxycarbonyl-Ser-Leu-Gly-Arg + 7-amino-4-methylcoumarin | - |
? | |
complement component C2 + H2O | the P1'-P4' substrate residues of C2 confer greater affinity of substrate for enzyme and also induce a sigmoidal dependence of enzyme velocity on substrate concentration. The substrate gives rise to homotropic positive cooperative behavior in the enzyme | Homo sapiens | complement component C2a + complement component C2b | - |
? | |
complement component C4 + H2O | the P1'-P4' substrate residues of C4 confer greater affinity of substrate for enzyme and also induce a sigmoidal dependence of enzyme velocity on substrate concentration. The substrate gives rise to homotropic positive cooperative behavior in the enzyme | Homo sapiens | complement component C4a + complement component C4b | - |
? | |
GLQRA + H2O | - |
Homo sapiens | GLQR + Ala | - |
? | |
GLQRAAEI + H2O | - |
Homo sapiens | GLQR + AAEI | - |
? | |
GLQRAEEI + H2O | - |
Homo sapiens | GLQR + AEEI | - |
? | |
GLQRAFEI + H2O | - |
Homo sapiens | GLQR + AFEI | - |
? | |
GLQRAHEI + H2O | - |
Homo sapiens | GLQR + AHEI | - |
? | |
GLQRAL + H2O | - |
Homo sapiens | GLQR + Ala-Leu | - |
? | |
GLQRALAI + H2O | - |
Homo sapiens | GLQR + ALAI | - |
? | |
GLQRALE + H2O | - |
Homo sapiens | GLQR + ALE | - |
? | |
GLQRALEA + H2O | - |
Homo sapiens | GLQR + ALEA | - |
? | |
GLQRALEE + H2O | - |
Homo sapiens | GLQR + ALEE | - |
? | |
GLQRALEF + H2O | - |
Homo sapiens | GLQR + ALEF | - |
? | |
GLQRALEH + H2O | - |
Homo sapiens | GLQR + ALEH | - |
? | |
GLQRALEI + H2O | - |
Homo sapiens | GLQR + ALEI | - |
? | |
GLQRALEK + H2O | - |
Homo sapiens | GLQR + ALEK | - |
? | |
GLQRALEL + H2O | - |
Homo sapiens | GLQR + ALEL | - |
? | |
GLQRALEM + H2O | - |
Homo sapiens | GLQR + ALEM | - |
? | |
GLQRALEP + H2O | - |
Homo sapiens | GLQR + ALEP | - |
? | |
GLQRALEQ + H2O | - |
Homo sapiens | GLQR + ALEQ | - |
? | |
GLQRALET + H2O | - |
Homo sapiens | GLQR + ALET | - |
? | |
GLQRALFI + H2O | - |
Homo sapiens | GLQR + ALFI | - |
? | |
GLQRALHI + H2O | - |
Homo sapiens | GLQR + ALHI | - |
? | |
GLQRALKI + H2O | - |
Homo sapiens | GLQR + ALKI | - |
? | |
GLQRALLI + H2O | - |
Homo sapiens | GLQR + ALLI | - |
? | |
GLQRALMI + H2O | - |
Homo sapiens | GLQR + ALMI | - |
? | |
GLQRALPI + H2O | - |
Homo sapiens | GLQR + ALPI | - |
? | |
GLQRALQI + H2O | - |
Homo sapiens | GLQR + ALQI | - |
? | |
GLQRALTI + H2O | - |
Homo sapiens | GLQR + ALTI | - |
? | |
GLQRAMEI + H2O | - |
Homo sapiens | GLQR + AMEI | - |
? | |
GLQRAPEI + H2O | - |
Homo sapiens | GLQR + APEI | - |
? | |
GLQRAQEI + H2O | - |
Homo sapiens | GLQR + AQEI | - |
? | |
GLQRATEI + H2O | - |
Homo sapiens | GLQR + ATEI | - |
? | |
GLQRELEI + H2O | - |
Homo sapiens | GLQR + ELEI | - |
? | |
GLQRFLEI + H2O | - |
Homo sapiens | GLQR + FLEI | - |
? | |
GLQRHLEI + H2O | - |
Homo sapiens | GLQR + HLEI | - |
? | |
GLQRKLEI + H2O | - |
Homo sapiens | GLQR + KLEI | - |
? | |
GLQRLLEI + H2O | - |
Homo sapiens | GLQR + LLEI | - |
? | |
GLQRMLEI + H2O | - |
Homo sapiens | GLQR + MLEI | - |
? | |
GLQRQLEI + H2O | - |
Homo sapiens | GLQR + QLEI | - |
? | |
GLQRTLEI + H2O | - |
Homo sapiens | GLQR + TLEI | - |
? | |
additional information | importance of the prime subsites of the C1s protease for recognition of substrates no cleavage of GLQRPLEI and GLQRAKEI | Homo sapiens | ? | - |
? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0000189 | - |
GLQRAPEI | pH 7.4, 37°C | Homo sapiens | |
0.0000205 | - |
GLQRELEI | pH 7.4, 37°C | Homo sapiens | |
0.0000394 | - |
GLQRA | pH 7.4, 37°C | Homo sapiens | |
0.0000421 | - |
GLQRAEEI | pH 7.4, 37°C | Homo sapiens | |
0.0000702 | - |
GLQRLLEI | pH 7.4, 37°C | Homo sapiens | |
0.0000702 | - |
GLQRQLEI | pH 7.4, 37°C | Homo sapiens | |
0.0000762 | - |
GLQRKLEI | pH 7.4, 37°C | Homo sapiens | |
0.0000978 | - |
GLQRALEL | pH 7.4, 37°C | Homo sapiens | |
0.0000978 | - |
GLQRALEQ | pH 7.4, 37°C | Homo sapiens | |
0.0000978 | - |
GLQRALEE | pH 7.4, 37°C | Homo sapiens | |
0.000119 | - |
GLQRAMEI | pH 7.4, 37°C | Homo sapiens | |
0.000136 | - |
GLQRALKI | pH 7.4, 37°C | Homo sapiens | |
0.000147 | - |
GLQRATEI | pH 7.4, 37°C | Homo sapiens | |
0.000155 | - |
GLQRFLEI | pH 7.4, 37°C | Homo sapiens | |
0.000169 | - |
GLQRAAEI | pH 7.4, 37°C | Homo sapiens | |
0.000171 | - |
GLQRALEM | pH 7.4, 37°C | Homo sapiens | |
0.000183 | - |
GLQRAQEI | pH 7.4, 37°C | Homo sapiens | |
0.000205 | - |
GLQRALEI | pH 7.4, 37°C | Homo sapiens | |
0.00021 | - |
2-aminobenzoyl-Gly-Leu-Gln-Arg-Ala-Leu-Glu-Ile-Lys(dinitrophenyl)-NH2 | pH 7.4, 37°C | Homo sapiens | |
0.00022 | - |
GLQRALEF | pH 7.4, 37°C | Homo sapiens | |
0.000239 | - |
GLQRMLEI | pH 7.4, 37°C | Homo sapiens | |
0.000244 | - |
GLQRALEH | pH 7.4, 37°C | Homo sapiens | |
0.000319 | - |
GLQRALE | pH 7.4, 37°C | Homo sapiens | |
0.000323 | - |
GLQRAQEI | pH 7.4, 37°C | Homo sapiens | |
0.00033 | - |
GLQRAFEI | pH 7.4, 37°C | Homo sapiens | |
0.000392 | - |
GLQRALEA | pH 7.4, 37°C | Homo sapiens | |
0.000415 | - |
GLQRHLEI | pH 7.4, 37°C | Homo sapiens | |
0.00044 | - |
GLQRALET | pH 7.4, 37°C | Homo sapiens | |
0.000683 | - |
GLQRAL | pH 7.4, 37°C | Homo sapiens | |
0.000807 | - |
GLQRALEP | pH 7.4, 37°C | Homo sapiens | |
0.000867 | - |
GLQRALEK | pH 7.4, 37°C | Homo sapiens | |
0.00139 | - |
2-aminobenzoyl -Ser-Leu-Gly-Arg-Lys-Ile-Gln-Ile-Lys(dinitrophenyl)-NH2 | pH 7.4, 37°C | Homo sapiens | |
0.00155 | - |
GLQRTLEI | pH 7.4, 37°C | Homo sapiens | |
0.00227 | - |
GLQRALMI | pH 7.4, 37°C | Homo sapiens | |
0.00232 | - |
GLQRAQEI | pH 7.4, 37°C | Homo sapiens | |
0.00244 | - |
GLQRALPI | pH 7.4, 37°C | Homo sapiens | |
0.00274 | - |
GLQRALAI | pH 7.4, 37°C | Homo sapiens | |
0.00279 | - |
GLQRALTI | pH 7.4, 37°C | Homo sapiens | |
0.00288 | - |
GLQRALFI | pH 7.4, 37°C | Homo sapiens | |
0.00296 | - |
GLQRALLI | pH 7.4, 37°C | Homo sapiens | |
0.00821 | - |
GLQRALHI | pH 7.4, 37°C | Homo sapiens | |
0.38 | - |
benzyloxycarbonyl-Gly-Leu-Gln-Arg-4-methylcoumaryl-7-amide | pH 7.4, 37°C | Homo sapiens | |
0.5 | - |
benzyloxycarbonyl-Ser-Leu-Gly-Arg-4-methylcoumaryl-7-amide | pH 7.4, 37°C | Homo sapiens |