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BRENDA support

Literature summary for 3.4.21.34 extracted from

  • Phipps, J.A.; Clermont, A.C.; Sinha, S.; Chilcote, T.J.; Bursell, S.E.; Feener, E.P.
    Plasma kallikrein mediates angiotensin II type 1 receptor-stimulated retinal vascular permeability (2009), Hypertension, 53, 175-181.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
1-benzyl-1H-pyrazole-4-carboxylic acid 4-carbamimidoyl-benzylamide ASP-440, small molecule inhibitor of plasma kallikrein Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
kininogen + H2O Rattus norvegicus
-
bradykinin + ?
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Rattus norvegicus

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
kininogen + H2O
-
Rattus norvegicus bradykinin + ?
-
?