Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Glp-Asn-Pro-D-Tyr-D-Trp-7-amido-4-methyl-coumarin | - |
Rattus norvegicus | |
Glp-Asn-Pro-D-Tyr-D-Trp-D-Trp-7-amido-4-methyl-coumarin | - |
Rattus norvegicus | |
Glp-Asn-Pro-D-Tyr-D-TrpNH2 | potent inhibitor of TRH-DE. Competetive, fully reversible and not time dependent inhibition | Rattus norvegicus | |
Glp-Asn-Pro-Tyr-Trp-7-amido-4-methyl-coumarin | - |
Rattus norvegicus | |
Glp-Asn-Pro-Tyr-Trp-Trp-7-amido-4-methyl-coumarin | - |
Rattus norvegicus | |
Glp-Asn-Pro-Tyr-TrpNH2 | - |
Rattus norvegicus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.035 | - |
thyrotropin-releasing hormone | - |
Rattus norvegicus | |
0.5 | - |
(3-Me-His2)thyrotropin-releasing hormone | - |
Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
male Wistar rats | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Rattus norvegicus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
(3-Me-His2)thyrotropin-releasing hormone + H2O | - |
Rattus norvegicus | ? | - |
? | |
thyrotropin-releasing hormone + H2O | - |
Rattus norvegicus | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
TRH-DE | - |
Rattus norvegicus |
TRH-degrading ectoenzyme | - |
Rattus norvegicus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000001 | - |
Glp-Asn-Pro-Tyr-Trp-Trp-7-amido-4-methyl-coumarin | - |
Rattus norvegicus | |
0.000029 | - |
Glp-Asn-Pro-D-Tyr-D-Trp-D-Trp-7-amido-4-methyl-coumarin | - |
Rattus norvegicus | |
0.000038 | - |
Glp-Asn-Pro-Tyr-Trp-7-amido-4-methyl-coumarin | - |
Rattus norvegicus | |
0.000096 | - |
Glp-Asn-Pro-D-Tyr-D-Trp-7-amido-4-methyl-coumarin | - |
Rattus norvegicus | |
0.000151 | - |
Glp-Asn-Pro-D-Tyr-D-TrpNH2 | - |
Rattus norvegicus | |
0.00064 | - |
Glp-Asn-Pro-Tyr-TrpNH2 | - |
Rattus norvegicus |