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BRENDA support

Literature summary for 3.4.14.5 extracted from

  • Edgerton, D.S.; Johnson, K.M.; Neal, D.W.; Scott, M.; Hobbs, C.H.; Zhang, X.; Duttaroy, A.; Cherrington, A.D.
    Inhibition of dipeptidyl peptidase-4 by vildagliptin during glucagon-like peptide 1 infusion increases liver glucose uptake in the conscious dog (2009), Diabetes, 58, 243-249.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
vildagliptin complete inhibition over 4 h after treatment with a single oral dose of 1 mg/kg vildagliptin Canis lupus familiaris

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
glucagon-like peptide 1 + H2O Canis lupus familiaris
-
?
-
?

Organism

Organism UniProt Comment Textmining
Canis lupus familiaris
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
blood plasma
-
Canis lupus familiaris
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
glucagon-like peptide 1 + H2O
-
Canis lupus familiaris ?
-
?
Gly-L-Pro-7-amido-4-methylcoumarin + H2O
-
Canis lupus familiaris Gly-L-Pro + 7-amino-4-methylcoumarin
-
?

Synonyms

Synonyms Comment Organism
dipeptidyl peptidase-4
-
Canis lupus familiaris
DPP-4
-
Canis lupus familiaris