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Literature summary for 3.4.14.5 extracted from

  • Gao, Y.D.; Feng, D.; Sheridan, R.P.; Scapin, G.; Patel, S.B.; Wu, J.K.; Zhang, X.; Sinha-Roy, R.; Thornberry, N.A.; Weber, A.E.; Biftu, T.
    Modeling assisted rational design of novel, potent, and selective pyrrolopyrimidine DPP-4 inhibitors (2007), Bioorg. Med. Chem. Lett., 17, 3877-3879.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
sitagliptin
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens P27487
-
-

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.000018
-
-
Homo sapiens sitagliptin