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BRENDA support

Literature summary for 3.4.11.2 extracted from

  • Gabrilovac, J.; Breljak, D.; Cupic, B.
    Regulation of aminopeptidase N (EC 3.4.11.2; APN; CD13) on the HL-60 cell line by TGF-beta1 (2008), Int. Immunopharmacol., 8, 613-623.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
transforming growth factor-beta1 transforming growth factor-beta1 at physiological concentrations (0.16 to 2.5 ng/ml) increases expression of CD13 both at mRNA and membrane protein level in a time- and concentration-dependent manner, increased membrane CD13 expression is associated with an increase of its enzyme activity, actinomycin-D abrogates the transforming growth factor-beta1-induced up-regulation of CD13 Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
membrane
-
Homo sapiens 16020
-

Metals/Ions

Metals/Ions Comment Organism Structure
Zn2+ dependent on Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
HL-60 cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
L-Ala-p-nitroanilide + H2O
-
Homo sapiens L-Ala + p-nitroaniline
-
?

Synonyms

Synonyms Comment Organism
aminopeptidase N
-
Homo sapiens
APN
-
Homo sapiens
CD13
-
Homo sapiens