Crystallization (Comment) | Organism |
---|---|
modeling of docking of 3-galloylamido-N-substituted-2,6-piperidinedione-N-acetamide inhibitors | Sus scrofa |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
bestatin | - |
Sus scrofa | |
N-((3S)-1-[2-(hydroxyamino)-2-oxoethyl]-2,6-dioxopiperidin-3-yl)-3,4,5-trimethoxybenzamide | - |
Sus scrofa | |
N-((3S)-1-[2-(methylhistidinyl)-2-oxoethyl]-2,6-dioxopiperidin-3-yl)-3,4,5-trimethoxybenzamide | - |
Sus scrofa |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
microsome | - |
Sus scrofa | - |
- |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Sus scrofa | - |
commercial preparation | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
kidney | - |
Sus scrofa | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
L-Leu-4-nitroanilide + H2O | - |
Sus scrofa | L-Leu + 4-nitroaniline | - |
? |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0024 | - |
pH 7.2, 37°C | Sus scrofa | bestatin | |
0.0031 | - |
pH 7.2, 37°C | Sus scrofa | N-((3S)-1-[2-(hydroxyamino)-2-oxoethyl]-2,6-dioxopiperidin-3-yl)-3,4,5-trimethoxybenzamide | |
0.0052 | - |
pH 7.2, 37°C | Sus scrofa | N-((3S)-1-[2-(methylhistidinyl)-2-oxoethyl]-2,6-dioxopiperidin-3-yl)-3,4,5-trimethoxybenzamide |