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Literature summary for 3.4.11.2 extracted from

  • Jardinaud, F.; Banisadr, G.; Noble, F.; Melik-Parsadaniantz, S.; Chen, H.; Dugave, C.; Laplace, H.; Rostene, W.; Fournie-Zaluski, M.C.; Roques, B.P.; Popovici, T.
    Ontogenic and adult whole body distribution of aminopeptidase N in rat investigated by in vitro autoradiography (2004), Biochimie, 86, 105-113.
    View publication on PubMed

Application

Application Comment Organism
medicine the enzyme might be a therapeutic target in pathological processes, such as tumor proliferation and/or angiogenesis associated with cancer development Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
2(S)-benzyl-3-[hydroxy(1'(R)-aminoethyl)phosphinyl]propanoyl-L-3-iodotyrosine iodinated RB129 Rattus norvegicus
RB129
-
Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Rattus norvegicus the enzyme is involved in hematopoiesis and bone growth, increased enzyme expression occurs during angiogenesis associated with cancer development ?
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
Wistar rats
-

Source Tissue

Source Tissue Comment Organism Textmining
bone adult Rattus norvegicus
-
cartilage
-
Rattus norvegicus
-
embryo
-
Rattus norvegicus
-
eye
-
Rattus norvegicus
-
heart
-
Rattus norvegicus
-
intestine
-
Rattus norvegicus
-
kidney
-
Rattus norvegicus
-
liver
-
Rattus norvegicus
-
lung
-
Rattus norvegicus
-
additional information ontogenic and adult whole body distribution of aminopeptidase N, developmental expression pattern in organ compartments, detailed overview Rattus norvegicus
-
pancreas adult Rattus norvegicus
-
rectum adult Rattus norvegicus
-
sense organ
-
Rattus norvegicus
-
spleen adult Rattus norvegicus
-
thymus
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information the enzyme is involved in hematopoiesis and bone growth, increased enzyme expression occurs during angiogenesis associated with cancer development Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
aminopeptidase N
-
Rattus norvegicus
APN
-
Rattus norvegicus