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Literature summary for 3.1.6.2 extracted from
- Design, synthesis, and biological evaluation of new arylamide derivatives possessing sulfonate or sulfamate moieties as steroid sulfatase enzyme inhibitors (2016), Bioorg. Med. Chem., 24, 2762-2767 .
Inhibitors
| Inhibitors | Comment | Organism | Structure |
|---|---|---|---|
| 4-(cyclohexanecarboxamido)phenyl sulfamate | 55.7% inhibition of isolated enzyme at 0.01 mM, 86.1% inhibition of the STS activity of JEG-3 carcinoma cells at 0.010 mM | Homo sapiens |  |
Organism
| Organism | UniProt | Comment | Textmining |
|---|---|---|---|
| Homo sapiens | P08842 | - |
- |
Source Tissue
| Source Tissue | Comment | Organism | Textmining |
|---|---|---|---|
| JEG-3 cell | placental carcinoma cell | Homo sapiens | - |
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Release 2023.1 (January 2023)
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