Inhibitors | Comment | Organism | Structure |
---|---|---|---|
amentoflavone | IC50: 0.0117 mM | Homo sapiens | |
bilobetin | IC50: 0.00152 mM | Homo sapiens | |
ginkgetin | IC50: 0.00059 mM | Homo sapiens | |
additional information | Gingko biloba dimeric flavonoids inhibit the cGMP-specific PDE5A1 | Homo sapiens | |
sciadopitysin | IC50: 0.00324 mM | Homo sapiens | |
sequoiaflavone | IC50: 0.0199 mM | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
recombinant PDE5A1 | - |
Synonyms | Comment | Organism |
---|---|---|
cGMP-phosphodiesterase-5 | - |
Homo sapiens |
PDE5A1 | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00059 | - |
IC50: 0.00059 mM | Homo sapiens | ginkgetin | |
0.00152 | - |
IC50: 0.00152 mM | Homo sapiens | bilobetin | |
0.00324 | - |
IC50: 0.00324 mM | Homo sapiens | sciadopitysin | |
0.0117 | - |
IC50: 0.0117 mM | Homo sapiens | amentoflavone | |
0.0199 | - |
IC50: 0.0199 mM | Homo sapiens | sequoiaflavone |