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Literature summary for 3.1.4.35 extracted from

  • Bosgraaf, L.; Russcher, H.; Snippe, H.; Bader, S.; Wind, J.; Van Haastert, P.J.M.
    Identification and characterization of two unusual cGMP-stimulated phosphodiesterases in Dictyostelium (2002), Mol. Biol. Cell, 13, 3878-3889.
    View publication on PubMedView publication on EuropePMC

Activating Compound

Activating Compound Comment Organism Structure
8-bromo-cGMP
-
Dictyostelium
cGMP maximal 2.4fold activation below 0.001 mM, half-maximal activation at 0.00016 mM, inhibition above 0.001 mM Dictyostelium

Inhibitors

Inhibitors Comment Organism Structure
cAMP inhibition at high concentrations Dictyostelium
cGMP inhibition above 0.001 mM Dictyostelium

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.0052
-
cGMP
-
Dictyostelium

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
guanosine 3',5'-cyclic phosphate + H2O Dictyostelium
-
guanosine 5'-phosphate
-
?

Organism

Organism UniProt Comment Textmining
Dictyostelium
-
strains AX3 and DH1
-

Purification (Commentary)

Purification (Comment) Organism
partially purified Dictyostelium

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
guanosine 3',5'-cyclic phosphate + H2O
-
Dictyostelium guanosine 5'-phosphate
-
?

Synonyms

Synonyms Comment Organism
cGMP-stimulated phosphodiesterase
-
Dictyostelium
GbpA
-
Dictyostelium

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
1.8
-
cAMP
-
Dictyostelium