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Literature summary for 3.1.4.17 extracted from

  • Mukai, J.; Asai, T.; Naka, M.; Tanaka, T.
    Separation and characterization of a novel isoenzyme of cyclic nucleotide phosphodiesterase from rat cerebrum (1994), Br. J. Pharmacol., 111, 389-390.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
nicardipine weak inhibitor Rattus norvegicus
rolipram weak inhibitor Rattus norvegicus
SKF 94120 weak inhibitor Rattus norvegicus
zaprinast weak inhibitor Rattus norvegicus

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information three isoenzymes Rattus norvegicus

Localization

Localization Comment Organism GeneOntology No. Textmining
cytosol
-
Rattus norvegicus 5829
-

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
telencephalon
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3',5'-cAMP + H2O
-
Rattus norvegicus 5'-AMP
-
?
3',5'-cGMP + H2O
-
Rattus norvegicus 5'-GMP
-
?
nucleoside 3',5'-cyclic phosphate + H2O
-
Rattus norvegicus nucleoside 5'-phosphate
-
?