Inhibitors | Comment | Organism | Structure |
---|---|---|---|
aflatoxin B1 | 50% inhibition at 0.031 mM by increase of Km-value and decrease of vmax-value. Partial recativation by 2-aldoxime, i.e. 2-PAM, pyridin-2-aldoxime 1-methoiodide | Mus musculus | |
BW284c51 | 50% inhibition at 0.000021 mM | Mus musculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.04 | - |
acetylthiocholine | pH 7.2, 25°C | Mus musculus | |
0.062 | - |
acetylthiocholine | pH 7.2, 25°C, presence of aflatoxin B1 at 0.001 mM | Mus musculus | |
0.133 | - |
acetylthiocholine | pH 7.2, 25°C, presence of aflatoxin B1 at 0.1 mM | Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | - |
isoforms G1 and G4 | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Mus musculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
acetylthiocholine + H2O | - |
Mus musculus | acetate + thiocholine | - |
? |