Inhibitors | Comment | Organism | Structure |
---|---|---|---|
4-bromophenacyl bromide | alkylation with 4-bromophenacyl bromide leads to the complete loss of its enzymatic activity signifying the crucial role of histidine residue in catalysis | Daboia russelii |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
13597 | - |
electrospray ionization mass spectrometry | Daboia russelii |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Daboia russelii | C0HK16 | - |
- |
Purification (Comment) | Organism |
---|---|
- |
Daboia russelii |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
venom | - |
Daboia russelii | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
1,2-diheptanoylthio-phosphatidylcholine + H2O | - |
Daboia russelii | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
Daboxin P | - |
Daboia russelii |
Temperature Stability Minimum [°C] | Temperature Stability Maximum [°C] | Comment | Organism |
---|---|---|---|
72 | - |
Tm value is 71.59°C | Daboia russelii |
pH Stability | pH Stability Maximum | Comment | Organism |
---|---|---|---|
3 | - |
stable at | Daboia russelii |
7 | - |
stable at | Daboia russelii |
General Information | Comment | Organism |
---|---|---|
physiological function | the crude venom of Daboia r. russelii has prominent cytotoxic effect on HEK-293 and MCF-7 cells in a dose dependent manner. Phospholipase A2 enzyme from Indian viper (Daboia russelii russelii) venom targets both factor X and factor Xa for its anticoagulant activity | Daboia russelii |