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Literature summary for 3.1.1.13 extracted from

  • Chiou, S.Y.; Lin, M.C.; Hwang, M.T.; Chang, H.G.; Lin, G.
    Benzene-di-N-substituted carbamates as conformationally constrained substrate analogs of cholesterol esterase (2008), Protein J., 27, 276-282.
    View publication on PubMed
Search for more literature for 3.1.1.13

Inhibitors

Inhibitors Comment Organism Structure
benzene-1,2-di-N-benzylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,2-di-N-n-butylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,2-di-N-n-hexylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,2-di-N-n-octylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,2-di-N-t-butylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,3-di-N-benzylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,3-di-N-n-butylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,3-di-N-n-hexylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,3-di-N-n-octylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,3-di-N-t-butylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,4-di-N-benzylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,4-di-N-n-butylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,4-di-N-n-hexylcarbamate pseudo substrate inhibitor Sus scrofa
benzene-1,4-di-N-octylcarbamates pseudo substrate inhibitor Sus scrofa
benzene-1,4-di-N-t-butylcarbamate pseudo substrate inhibitor Sus scrofa

Organism

Organism UniProt Comment Textmining
Sus scrofa
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
pancreas
-
 Sus scrofa
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
p-nitrophenyl butyrate + H2O
-
 Sus scrofa p-nitrophenol + butyrate
-
 ?

Synonyms

Synonyms Comment Organism
CEase
-
 Sus scrofa
cholesterol esterase
-
 Sus scrofa

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.0004
-
 benzene-1,3-di-N-n-octylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.0007
-
 benzene-1,4-di-N-n-octylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.001
-
 benzene-1,3-di-N-n-hexylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.0012
-
 benzene-1,3-di-N-n-butylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.0012
-
 benzene-1,4-di-N-n-hexylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.0016
-
 benzene-1,3-di-N-t-butylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.0017
-
 benzene-1,3-di-N-benzylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.0018
-
 benzene-1,4-di-N-n-butylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.002
-
 benzene-1,4-di-N-t-butylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.004
-
 benzene-1,2-di-N-benzylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.005
-
 benzene-1,4-di-N-benzylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.007
-
 benzene-1,2-di-N-n-octylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.02
-
 benzene-1,2-di-N-n-hexylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.027
-
 benzene-1,2-di-N-n-butylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa
0.03
-
 benzene-1,2-di-N-t-butylcarbamate in sodium phosphate buffer (0.1 M, pH 7.0), at 25°C Sus scrofa