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Literature summary for 2.7.11.13 extracted from

  • Meng, Z.; Bischof, J.; Ianes, C.; Henne-Bruns, D.; Xu, P.; Knippschild, U.
    CK1delta kinase activity is modulated by protein kinase C alpha (PKCalpha)-mediated site-specific phosphorylation (2016), Amino Acids, 48, 1185-1197.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
Go-6983 isoform PKCalpha-specific inhibitor Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + casein kinase 1delta Homo sapiens phosphorylation at Ser328, Thr329, and Ser370 ADP + phosphorylated casein kinase 1delta
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
COLO-357 cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + casein kinase 1delta phosphorylation at Ser328, Thr329, and Ser370 Homo sapiens ADP + phosphorylated casein kinase 1delta
-
?

Synonyms

Synonyms Comment Organism
PKCalpha
-
Homo sapiens
protein kinase C alpha
-
Homo sapiens