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Literature summary for 2.7.11.12 extracted from

  • Munhoz, C.D.; Kawamoto, E.M.; de Sa Lima, L.; Lepsch, L.B.; Glezer, I.; Marcourakis, T.; Scavone, C.
    Glutamate modulates sodium-potassium-ATPase through cyclic GMP and cyclic GMP-dependent protein kinase in rat striatum (2005), Cell Biochem. Funct., 23, 115-123.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
8-bromo-cGMP
-
Rattus norvegicus
cGMP level is increased by NO and glutamate Rattus norvegicus
additional information glutamate induced NO, and increased NO release from sodium nitroprusside and S-nitroso-N-acetylpenicillamine increase cGMP level which increases PKG activity, overview Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
KT5823 specific for PKG Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + Na+/K+ ATPase Rattus norvegicus the enzyme has a positive regulatory function on the ion pump activity induced by No and glutamate via increased cGMP, overview ADP + phosphorylated Na+/K+ ATPase
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
male Wistar rats
-

Source Tissue

Source Tissue Comment Organism Textmining
corpus striatum
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + Na+/K+ ATPase
-
Rattus norvegicus ADP + phosphorylated Na+/K+ ATPase
-
?
ATP + Na+/K+ ATPase the enzyme has a positive regulatory function on the ion pump activity induced by No and glutamate via increased cGMP, overview Rattus norvegicus ADP + phosphorylated Na+/K+ ATPase
-
?

Synonyms

Synonyms Comment Organism
PKG
-
Rattus norvegicus

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
34
-
assay at, in vivo Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.4
-
assay at, in vivo Rattus norvegicus

Cofactor

Cofactor Comment Organism Structure
ATP
-
Rattus norvegicus