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BRENDA support

Literature summary for 2.7.11.11 extracted from

  • Grueb, M.; Bartz-Schmidt, K.U.; Rohrbach, J.M.
    Adrenergic regulation of cAMP/protein kinase A pathway in corneal epithelium and endothelium (2008), Ophthalmic Res., 40, 322-328.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
additional information beta-adrenergic stimulation with isoprenaline leads to activation of PKA via stimulation of adenylyl cyclase Bos taurus

Inhibitors

Inhibitors Comment Organism Structure
additional information alpha2A-adrenoceptor stimulation with brimonidine inhibits PKA activity via inhibition of adenylyl cyclase Bos taurus

Organism

Organism UniProt Comment Textmining
Bos taurus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
corneal epithelium
-
Bos taurus
-
endothelium
-
Bos taurus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + Kemptide
-
Bos taurus ADP + Kemptide phosphate
-
?

Synonyms

Synonyms Comment Organism
PKA
-
Bos taurus
protein kinase A
-
Bos taurus

Cofactor

Cofactor Comment Organism Structure
ATP
-
Bos taurus
cAMP dependent Bos taurus