Activating Compound | Comment | Organism | Structure |
---|---|---|---|
cAMP | - |
Oryctolagus cuniculus | |
cBIMPS | - |
Oryctolagus cuniculus | |
forskolin | activates at concentration above 0.001 mM | Oryctolagus cuniculus | |
isoproterenol | at concentration below 0.001 mM | Oryctolagus cuniculus | |
Vasoactive intestinal peptide | i.e. VIP | Oryctolagus cuniculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
myristoylated PKI14-22 amide | selective peptide inhibitor of P KA | Oryctolagus cuniculus |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | - |
Oryctolagus cuniculus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Oryctolagus cuniculus | inositol 1,4,5-trisphosphate receptor-I is no substrate of PKA in vivo | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Oryctolagus cuniculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
smooth muscle cell | gastric, primary | Oryctolagus cuniculus | - |
stomach | - |
Oryctolagus cuniculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + inositol 1,4,5-trisphosphate receptor-I | isolated catalytic subunit of PKA, selective phosphorylation at Ser1589 and Ser1755 | Oryctolagus cuniculus | ADP + phosphorylated inositol 1,4,5-trisphosphate receptor-I | - |
? | |
additional information | inositol 1,4,5-trisphosphate receptor-I is no substrate of PKA in vivo | Oryctolagus cuniculus | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PKA | - |
Oryctolagus cuniculus |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
31 | - |
in vivo phosphorylation assay at | Oryctolagus cuniculus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.4 | - |
assay at | Oryctolagus cuniculus |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
ATP | - |
Oryctolagus cuniculus |