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Literature summary for 2.7.11.10 extracted from

  • Tang, H.; Park, S.; Sun, S.C.; Trumbly, R.; Ren, G.; Tsung, E.; Yeung, K.C.
    RKIP inhibits NF-kappaB in cancer cells by regulating upstream signaling components of the IkappaB kinase complex (2010), FEBS Lett., 584, 662-668.
    View publication on PubMedView publication on EuropePMC

Activating Compound

Activating Compound Comment Organism Structure
TAK1 critical direct upsteam activating kinase of IKK Homo sapiens
TRAF6 upstream activator of IKK kinase complex Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + [IkappaB protein] Homo sapiens
-
ADP + [IkappaB phosphoprotein]
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
293-IL-1RI cell
-
Homo sapiens
-
A-549 cell
-
Homo sapiens
-
DU-145 cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + [IkappaB protein]
-
Homo sapiens ADP + [IkappaB phosphoprotein]
-
?

Subunits

Subunits Comment Organism
heterotrimer IkappaB kinase, IKK, consists of two catalytic subunits, IKKalpha and IKKbeta, and a regulatory subunit called NEMO or IKKgamma Homo sapiens

Synonyms

Synonyms Comment Organism
IkappaB kinase
-
Homo sapiens
IKK
-
Homo sapiens

Cofactor

Cofactor Comment Organism Structure
ATP
-
Homo sapiens