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Literature summary for 2.7.10.2 extracted from
- Development of potent inhibitors of receptor tyrosine kinases by ligand-based drug design and target-biased phenotypic screening (2018), J. Med. Chem., 61, 2104-2110 .
Inhibitors
| Inhibitors | Comment | Organism | Structure |
|---|---|---|---|
| BGB324 | i.e. Bemcentinib | Homo sapiens | |
| additional information | development of potent inhibitors of receptor tyrosine kinases by ligand-based drug design and target-biased phenotypic screening | Homo sapiens |
Organism
| Organism | UniProt | Comment | Textmining |
|---|---|---|---|
| Homo sapiens | P12931 | - |
- |
Synonyms
| Synonyms | Comment | Organism |
|---|---|---|
| Src kinase | - |
Homo sapiens |
IC50 Value
| IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
|---|---|---|---|---|---|
| 0.000037 | - |
pH and temperature not specified in the publication | Homo sapiens | BGB324 |
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Release 2023.1 (January 2023)
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