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Literature summary for 2.7.10.2 extracted from

  • Yamaoka, K.; Tanaka, Y.
    Jak inhibitor: possibility and mechanism as a new disease modifying anti-rheumatic drug (2009), Nihon Rinsho Meneki Gakkai Kaishi, 32, 85-91.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
CP690,550 targeting Jak3 Homo sapiens
INCB18424 targeting Jak1/2 Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + a [protein]-L-tyrosine Homo sapiens
-
ADP + a [protein]-L-tyrosine phosphate
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
dendritic cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + a [protein]-L-tyrosine
-
Homo sapiens ADP + a [protein]-L-tyrosine phosphate
-
?

Synonyms

Synonyms Comment Organism
Jak1
-
Homo sapiens
JAK2
-
Homo sapiens
Jak3
-
Homo sapiens
Janus kinase
-
Homo sapiens
Tyk2
-
Homo sapiens

Cofactor

Cofactor Comment Organism Structure
ATP
-
Homo sapiens