Activating Compound | Comment | Organism | Structure |
---|---|---|---|
additional information | Src is activated by mechanical stretch of beta1 integrin, cell swelling and integrin clustering | Oryctolagus cuniculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
4-amino-5-(4-chlorophenyl)-7-(tert-butyl)pyrazolo[3,4-d]pyrimidine | i.e. PP2, inhibits Src | Oryctolagus cuniculus | |
genistein | - |
Oryctolagus cuniculus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Oryctolagus cuniculus | Src activates an outwardly rectifying chloride current in myocytes being involved in osmotic swelling, enzyme inhibition also inhibits stretch-activated Cl- current, mechanism, overview | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Oryctolagus cuniculus | - |
New Zealand white rabbits | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
myocyte | left ventricular | Oryctolagus cuniculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Src activates an outwardly rectifying chloride current in myocytes being involved in osmotic swelling, enzyme inhibition also inhibits stretch-activated Cl- current, mechanism, overview | Oryctolagus cuniculus | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
Protein tyrosine kinase | - |
Oryctolagus cuniculus |
PTK | - |
Oryctolagus cuniculus |
Src | - |
Oryctolagus cuniculus |