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Literature summary for 2.7.10.2 extracted from

  • Ren, Z.; Baumgarten, C.M.
    Antagonistic regulation of swelling-activated Cl- current in rabbit ventricle by Src and EGFR protein tyrosine kinases (2005), Am. J. Physiol., 288, H2628-2636.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
4-amino-5-(4-chlorophenyl)-7-(tert-butyl)pyrazolo[3,4-d] pyrimidine i.e. pp2, inhibits Src family PTKs Oryctolagus cuniculus
genistein broad spectrum PTK inhibitor Oryctolagus cuniculus
additional information no inhibition of Src with pp3, i.e. 4-amino-7-phenylpyrazolo[3,4-d] pyrimidine Oryctolagus cuniculus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Oryctolagus cuniculus antagonistic regulation of swelling-activated Cl- current in rabbit ventricle by Src and EGFR protein tyrosine kinases, overview ?
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?

Organism

Organism UniProt Comment Textmining
Oryctolagus cuniculus
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New Zealand white rabbits
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Source Tissue

Source Tissue Comment Organism Textmining
heart
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Oryctolagus cuniculus
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myocyte ventricular, primary Oryctolagus cuniculus
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ventriculus left Oryctolagus cuniculus
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Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information antagonistic regulation of swelling-activated Cl- current in rabbit ventricle by Src and EGFR protein tyrosine kinases, overview Oryctolagus cuniculus ?
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?

Synonyms

Synonyms Comment Organism
Protein tyrosine kinase
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Oryctolagus cuniculus
PTK
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Oryctolagus cuniculus
Src
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Oryctolagus cuniculus