Cloned (Comment) | Organism |
---|---|
His-tag, expressed in Escherichia coli BL21(DE3)-pRIL | Plasmodium falciparum 3D7 |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2-amino-1-butanol | - |
Plasmodium falciparum 3D7 | |
hemicholinium-3 | - |
Plasmodium falciparum 3D7 | |
SAR97276 | - |
Plasmodium falciparum 3D7 |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
ethanolamine | above 500 mM | Plasmodium falciparum 3D7 | |
0.1353 | - |
choline | recombinant protein | Plasmodium falciparum 3D7 |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
52000 | - |
1 * 52000, gel filtration | Plasmodium falciparum 3D7 |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Plasmodium falciparum 3D7 | Q8IM71 | - |
- |
Purification (Comment) | Organism |
---|---|
- |
Plasmodium falciparum 3D7 |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
62.2 micromol/min/mg for ethanolamine | Plasmodium falciparum 3D7 |
10.8 | - |
recombinant protein | Plasmodium falciparum 3D7 |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
choline + ATP | - |
Plasmodium falciparum 3D7 | O-phosphocholine + ADP | - |
? |
Subunits | Comment | Organism |
---|---|---|
monomer | 1 * 52000, gel filtration | Plasmodium falciparum 3D7 |
Synonyms | Comment | Organism |
---|---|---|
choline kinase | - |
Plasmodium falciparum 3D7 |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.9 | - |
SAR97276 | calculated from Dixon analysis | Plasmodium falciparum 3D7 | |
1.03 | - |
SAR97276 | calculated from Lineweaver-Burk analysis | Plasmodium falciparum 3D7 |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.22 | - |
endogenous enzyme | Plasmodium falciparum 3D7 | hemicholinium-3 | |
0.52 | - |
endogenous enzyme | Plasmodium falciparum 3D7 | SAR97276 | |
0.58 | - |
recombinant enzyme | Plasmodium falciparum 3D7 | hemicholinium-3 | |
1.12 | - |
recombinant enzyme | Plasmodium falciparum 3D7 | SAR97276 | |
3.2 | - |
endogenous enzyme | Plasmodium falciparum 3D7 | 2-amino-1-butanol |