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Literature summary for 2.7.1.158 extracted from

  • Wundenberg, T.; Grabinski, N.; Lin, H.; Mayr, G.W.
    Discovery of InsP6-kinases as InsP6-dephosphorylating enzymes provides a new mechanism of cytosolic InsP6 degradation driven by the cellular ATP/ADP ratio (2014), Biochem. J., 462, 173-184.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
N2-(m-trifluoromethylbenzyl),N6-(p-nitrobenzyl)purine selective inhibitor Homo sapiens
N2-(m-trifluoromethylbenzyl),N6-(p-nitrobenzyl)purine selective inhibitor Rattus norvegicus

Localization

Localization Comment Organism GeneOntology No. Textmining
cytosol
-
Homo sapiens 5829
-
cytosol
-
Rattus norvegicus 5829
-
nucleus
-
Homo sapiens 5634
-
nucleus
-
Rattus norvegicus 5634
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + 1D-myo-inositol 1,3,4,5,6-pentakisphosphate Homo sapiens
-
ADP + 1D-myo-inositol hexakisphosphate
-
?
ATP + 1D-myo-inositol 1,3,4,5,6-pentakisphosphate Rattus norvegicus
-
ADP + 1D-myo-inositol hexakisphosphate
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
blood
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + 1D-myo-inositol 1,3,4,5,6-pentakisphosphate
-
Homo sapiens ADP + 1D-myo-inositol hexakisphosphate
-
?
ATP + 1D-myo-inositol 1,3,4,5,6-pentakisphosphate
-
Rattus norvegicus ADP + 1D-myo-inositol hexakisphosphate
-
?
additional information the enzyme changes its kinase activity towards 1D-myo-inositol hexakisphosphate at a decreasing ATP/ADP ratio to an ADP phosphotransferase activity and dephosphorylate 1D-myo-inositol hexakisphosphate Homo sapiens ?
-
?
additional information the enzyme changes its kinase activity towards 1D-myo-inositol hexakisphosphate at a decreasing ATP/ADP ratio to an ADP phosphotransferase activity and dephosphorylate 1D-myo-inositol hexakisphosphate Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
InsP6-kinase
-
Homo sapiens
InsP6-kinase
-
Rattus norvegicus
IP6K
-
Homo sapiens
IP6K
-
Rattus norvegicus