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Literature summary for 2.7.1.107 extracted from

  • Takahashi, N.; Nagamine, M.; Tanno, S.; Motomura, W.; Kohgo, Y.; Okumura, T.
    A diacylglycerol kinase inhibitor, R59022, stimulates glucose transport through a MKK3/6-p38 signaling pathway in skeletal muscle cells (2007), Biochem. Biophys. Res. Commun., 360, 244-250.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
R59022 specifc inhibitor of diacylglycerol kinase. Treatment significantly increases glucose transport, p38 and MKK3/6 activation in myotubes. The R59022-induced glucose transport is blocked by SB203580, a specific p38 inhibitor. R59022 fails to stimulate both possible known mechanisms to enhance glucose transport, an IRS1-PI3K-Akt pathway, muscle contraction signaling or GLUT1 and GLUT4 expression Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
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Source Tissue

Source Tissue Comment Organism Textmining
C2C12 cell
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Mus musculus
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myotube expression of diacylglycerol kinase isoform alpha, delta, epsilon, zeta, or theta mRNA Mus musculus
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