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Literature summary for 2.5.1.15 extracted from

  • Auliff, A.; Wilson, D.W.; Russell, B.; Gao, Q.; Chen, N.; Anh le, N.; Maguire, J.; Bell, D.; O'Neil, M.T.; Cheng, Q.
    Amino acid mutations in Plasmodium vivax DHFR and DHPS from several geographical regions and susceptibility to antifolate drugs (2006), Am. J. Trop. Med. Hyg., 75, 617-621.
    View publication on PubMed

Protein Variants

Protein Variants Comment Organism
additional information assessment of mutations in DHPS associated with antifolate resistance in several geographical regions Plasmodium vivax

Inhibitors

Inhibitors Comment Organism Structure
cycloguanil
-
Plasmodium vivax
pyrimethamine
-
Plasmodium vivax
WR99210
-
Plasmodium vivax

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
2-amino-4-hydroxy-6-hydroxymethyl-7,8-dihydropteridine diphosphate + 4-aminobenzoate Plasmodium vivax
-
diphosphate + 7,8-dihydropteroate
-
?

Organism

Organism UniProt Comment Textmining
Plasmodium vivax Q00LY0 fragment of dihydropteroate synthase
-

Source Tissue

Source Tissue Comment Organism Textmining
bloodstream form
-
Plasmodium vivax
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2-amino-4-hydroxy-6-hydroxymethyl-7,8-dihydropteridine diphosphate + 4-aminobenzoate
-
Plasmodium vivax diphosphate + 7,8-dihydropteroate
-
?

Synonyms

Synonyms Comment Organism
7,8-dihydropteroate synthase
-
Plasmodium vivax
DHPS
-
Plasmodium vivax
dihydropteroate synthetase
-
Plasmodium vivax
pvdhps
-
Plasmodium vivax